Search Result "SAR-activity"


Research Article

In silico Screening of Phytoconstituents with Antiviral Activities Against SARS-COV-2 Main Protease, Nsp12 Polymerase, and Nsp13 Helicase Proteins

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 0 Year: 2021 Page: 1-17
Author(s): Jainey James,Divya Jyothi,Sneh Priya

Short Communication

Does Hypofractionated Radiotherapy Regimens Increase the Vulnerability to SARS- COV-2 by Influencing ACE-2 Activity?

Journal: Coronaviruses
Volume: 2 Issue: 4 Year: 2021 Page: 419-421
Author(s): Ghofrane Salhi Cherkaoui,Sara Taleb,Youness Kadil,Houda Filali

Design, SAR, Angiogenic Activities Evaluation and Pro-Angiogenic Mechanism of New Marine Cyclopeptide Analogs

Journal: Current Medicinal Chemistry
Volume: 20 Issue: 9 Year: 2013 Page: 1183-1194
Author(s): J. Li,X. Lu,Q. Wu,G. Yu,Z. Xu,L. Qiu,Z. Pei,Y. Lin,J. Pang

SAR Modeling: Effect of Experimental Ambiguity

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 6 Issue: 2 Year: 2003 Page: 161-166
Author(s): Bhavani P. Thampatty, Herbert S. Rosenkranz

Research Article

Synthesis and SAR Study of Simple Aryl Oximes and Nitrofuranyl Derivatives with Potent Activity Against Mycobacterium tuberculosis

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 1 Year: 2020 Page: 12-20
Author(s): Cristiane França da Costa,Marcus Vinicius Nora de Souza,Maria Cristina da Silva Lourenço,Elaine Soares Coimbra,Guilherme da Silva Lourenço Carvalho,James Wardell,Stephane Lima Calixto,Juliana da Trindade Granato

Research Article

In Silico Insight into the Inhibitory Effects of Active Antidiabetic Compoundsfrom Medicinal Plants Against SARS-CoV-2 Replication and PosttranslationalModification

Journal: Coronaviruses
Volume: 3 Issue: 2 Year: 2022 Page: 70-79
Author(s): Habibu Tijjani,Adamu Idris Matinja,Ahmed Olatunde,Maryam Haladu Zangoma,Abubakar Mohammed,Muhammad Akram,Akinwunmi Oluwaseun Adeoye,Hamza Lawal

Recent Progress in Structure Activity Relationship and Mechanistic Studies of Taxol Analogues

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 5 Issue: 1 Year: 2005 Page: 1-12
Author(s): W.- S. Fang, X.- T. Liang

Novel High Throughput Polymer Biocompatibility Screening Designed for SAR (Structure-Activity Relationship): Application for Evaluating Polymer Coatings for Cardiovascular Drug-Eluting Stents

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 12 Issue: 7 Year: 2009 Page: 664-676
Author(s): Ayala Hezi-Yamit, Carol Sullivan, Jennifer Wong, Laura David, Mingfei Chen, Peiwen Cheng, David Shumaker, Josiah Wilcox, Kishore Udipi

Benzenecarboxamide Analogs of Fluoroquinolones (BCFQs). Antibacterial Activity and SAR Studies

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 2 Year: 2006 Page: 108-111
Author(s): M. J. Nieto, F. L. Alovero, R. H. Manzo, M. R. Mazzieri

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