Search Result "COX-2 enzyme."


Research Article

3D-QSAR and Molecular Docking Studies on Oxadiazole Substituted Benzimidazole Derivatives: Validation of Experimental Inhibitory Potencies Towards COX-2

Journal: Current Computer-Aided Drug Design
Volume: 15 Issue: 4 Year: 2019 Page: 277-293
Author(s): Vivek Asati,Piyush Ghode,Shalini Bajaj,Sanmati K. Jain,Sanjay K. Bharti

Research Article

Molecular Dynamics Studies on COX-2 Protein-tyrosine Analogue Complex and Ligand-based Computational Analysis of Halo-substituted Tyrosine Analogues

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 1 Year: 2019 Page: 1211-1232
Author(s): Ayarivan Puratchikody,Appavoo Umamaheswari,Navabshan Irfan,Dharmarajan Sriram

Research Article

Synthesis of 1,3-benzoxazines Based on 2,4,4-trimethyl-7,2’,4’-trihydroxy Flavan: Antibacterial, Anti-inflammatory, Cyclooxygenase-2 Inhibition and Molecular Modelling Studies

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 1 Year: 2019 Page: 58-65
Author(s): Issam A. Mohammed,Mahmood Ahmed,Rabia Ikram,Muhammad Muddassar,Muhammad Abdul Qadir,Khalijah Binti Awang

Research Article

Application of a Validated QSTR Model for Repurposing COX-2 Inhibitor Coumarin Derivatives as Potential Antitumor Agents

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 1121-1128
Author(s): Gulcin Tugcu,Hande Sipahi,Ahmet Aydin

Research Article

Synthesis, Anti-inflammatory, Antimicrobial Potential and Molecular Docking Studies of 4,5-Disubstituted-1,2,4-Triazole Thioacetate Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 7 Year: 2019 Page: 734-745
Author(s): Muhammad Nouman Arif,Humaira Nadeem,Rehan Zafar Paracha,Arif-ullah Khan,Muhammad Imran,Fawad Ali

Review Article

Cyclooxygenase-2 Inhibitors as a Therapeutic Target in Inflammatory Diseases

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 1 Year: 2019 Page: 3225-3241
Author(s): Miguel D. Ferrer,Carla Busquets-Cortés,Xavier Capó,Silvia Tejada,Josep A. Tur,Antoni Pons,Antoni Sureda

Review Article

Celecoxib in Cancer Therapy and Prevention – Review

Journal: Current Drug Targets
Volume: 20 Issue: 3 Year: 2019 Page: 302-315
Author(s): Natalia Tołoczko-Iwaniuk,Dorota Dziemiańczyk-Pakieła,Beata Klaudia Nowaszewska,Katarzyna Celińska-Janowicz,Wojciech Miltyk

Research Article

Synthesis, Molecular Modelling and Antibacterial Activity Against Helicobacter pylori of Novel Diflunisal Derivatives as Urease Enzyme Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 4 Year: 2019 Page: 392-400
Author(s): Göknil Pelin Coşku,Teodora Djikic,Sadik Kalayci,Kemal Yelekci,Fikrettin Sahin,Ş. Güniz Küçükgüzel

Review Article

Neuroprotective Methodologies of Co-Enzyme Q10 Mediated Brain Hemorrhagic Treatment: Clinical and Pre-Clinical Findings

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 18 Issue: 6 Year: 2019 Page: 446-467
Author(s): Kajal Rajdev,Sidharth Mehan

Review Article

Potential Enzymatic Targets in Alzheimer’s: A Comprehensive Review

Journal: Current Drug Targets
Volume: 20 Issue: 3 Year: 2019 Page: 316-339
Author(s): Jahangir Alam,Lalit Sharma

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