Search Result "[11C]Tariquidar"


Substrates, Inhibitors and Activators of P-glycoprotein: Candidates for Radiolabeling and Imaging Perspectives

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1703-1714
Author(s): Nicola A. Colabufo, Francesco Berardi, Maria Grazia Perrone, Elena Capparelli, Mariangela Cantore, Carmela Inglese, Roberto Perrone

Evaluation of [11C]S14506 and [18F]S14506 in Rat and Monkey as Agonist PET Radioligands for Brain 5-HT1A Receptors

Journal: Current Radiopharmaceuticals
Volume: 3 Issue: 1 Year: 2010 Page: 9-18
Author(s): Shuiyu Lu, Jeih-San Liow, Sami S. Zoghbi, Jinsoo Hong, Robert B. Innis, Victor W. Pike

Carbon-11 Labeled Tracers for In Vivo Imaging of P-Glycoprotein Function: Kinetics, Advantages and Disadvantages

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1820-1833
Author(s): Gert Luurtsema, Joost Verbeek, Mark Lubberink, Adriaan A. Lammertsma, Rudi Dierckx, Philip Elsinga, Albert D. Windhorst, Aren van Waarde

Imaging of P-glycoprotein Function and Expression to Elucidate Mechanisms of Pharmacoresistance in Epilepsy

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1785-1791
Author(s): Wolfgang Loscher, Oliver Langer

Review Article

Kinetic Models for Measuring P-glycoprotein Function at the Blood-Brain Barrier with Positron Emission Tomography

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5786-5792
Author(s): Mark Lubberink

Current Frontiers

The Tetrahydroisoquinoline Scaffold in ABC Transporter Inhibitors that Act as Multidrug Resistance (MDR) Reversers

Journal: Current Topics in Medicinal Chemistry
Volume: 22 Issue: 31 Year: 2022 Page: 2535-2569
Author(s): Maria Novella Romanelli

Review Article

PET Tracers for Imaging of ABC Transporters at the Blood-Brain Barrier: Principles and Strategies

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5779-5785
Author(s): Gert Luurtsema,Philip Elsinga,Rudi Dierckx,Ronald Boellaard,Aren van Waarde

Review Article

Importance of P-gp PET Imaging in Pharmacology

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5830-5836
Author(s): Jun Toyohara

Review Article

Design and Synthesis of New Selective P-gp Substrates and Inhibitors

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5774-5778
Author(s): Mariangela Cantore,Marcello Leopoldo,Francesco Berardi,Roberto Perrone,Nicola Antonio Colabufo

PET and SPECT Radiotracers to Assess Function and Expression of ABC Transporters In Vivo

Journal: Current Drug Metabolism
Volume: 12 Issue: 8 Year: 2011 Page: 774-792
Author(s): Severin Mairinger, Thomas Erker, Markus Muller, Oliver Langer

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