Abstract
In recent years, pharmaceutical chemists have synthesized large numbers of andrographolide derivatives, which bear important biological activities such as anti-inflammatory, antibacterial, antivirus, antitumor, antidiabetic, and antifeedant. Consequently, corresponding SARs were increasingly obvious. This paper aimed to review all the available literature in this field, highlighting the significant achievements on the structural modification and SARs of andrographolide and its derivatives.
Keywords: Andrographolide derivatives, biological activities, SARs
Mini-Reviews in Medicinal Chemistry
Title:Biological Activities and Corresponding SARs of Andrographolide and Its Derivatives
Volume: 13 Issue: 2
Author(s): Bin Zhou, Dayong Zhang and Xiaoming Wu
Affiliation:
Keywords: Andrographolide derivatives, biological activities, SARs
Abstract: In recent years, pharmaceutical chemists have synthesized large numbers of andrographolide derivatives, which bear important biological activities such as anti-inflammatory, antibacterial, antivirus, antitumor, antidiabetic, and antifeedant. Consequently, corresponding SARs were increasingly obvious. This paper aimed to review all the available literature in this field, highlighting the significant achievements on the structural modification and SARs of andrographolide and its derivatives.
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Cite this article as:
Zhou Bin, Zhang Dayong and Wu Xiaoming, Biological Activities and Corresponding SARs of Andrographolide and Its Derivatives, Mini-Reviews in Medicinal Chemistry 2013; 13 (2) . https://dx.doi.org/10.2174/1389557511313020011
DOI https://dx.doi.org/10.2174/1389557511313020011 |
Print ISSN 1389-5575 |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-5607 |
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