Search Result "tyrosine kinase inhibitor"


Review Article

Recent Updates on the Therapeutic Potential of HER2 Tyrosine Kinase Inhibitors for the Treatment of Breast Cancer

Journal: Current Cancer Drug Targets
Volume: 18 Issue: 4 Year: 2018 Page: 306-327
Author(s): Heena Singla,Anjana Munshi,Raja Paramjit Singh Banipal,Vinod Kumar

Review Article

Development of Bruton’s Tyrosine Kinase Inhibitors for Rheumatoid Arthritis

Journal: Current Medicinal Chemistry
Volume: 25 Issue: 4 Year: 2018 Page: 5847-5859
Author(s): Jiahui Lv,Jingde Wu,Feng He,Ying Qu,Qiuqiong Zhang,Chenggong Yu

Review Article

Aurora Kinase Inhibitors in Head and Neck Cancer

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 3 Year: 2018 Page: 199-213
Author(s): Guangying Qi,Jing Liu,Sisi Mi,Takaaki Tsunematsu,Shengjian Jin,Wenhua Shao,Tian Liu,Naozumi Ishimaru,Bo Tang,Yasusei Kudo

Review Article

Genetic Polymorphism on the Pharmacokinetics and Pharmacodynamics of Plateletderived Growth Factor Receptor (PDGFR) Kinase Inhibitors

Journal: Current Drug Metabolism
Volume: 19 Issue: 1 Year: 2018 Page: 1168-1181
Author(s): Yi Qian,Lei Yu,Xue-Hui Zhang,Zi-Qing Yun Yuan,Ping Zhao,Lu-Ning Sun,Yong-Qing Wang

Research Article

Novel Tetrahydrobenzo [b] Thiophene Compounds Exhibit Anticancer Activity through Enhancing Apoptosis and Inhibiting Tyrosine Kinase

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 1761-1769
Author(s): Souad A. El-Metwally,Ali K. Khalil,Abeer M. El-Naggar,Wael M. El-Sayed

Research Article

3D-QSAR Studies on New Benzothiazole-Based Dual Functional Inhibitors of BCR-ABL Kinase Including the T315I Mutant

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 1 Year: 2018 Page: 1046-1056
Author(s): Shunlai Li,Chaorui Ren,Chenghu Lu,Xiuxiu Li,Hongguang Du

Research Article

Heterocyclization of Thiophenes Derived from Estrone Followed by Cytotoxic, HTRF Kinase and Pim-1 Kinase Evaluations

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 1711-1728
Author(s): Mahmoud A. Abdelaziz Mahmoud,Rafat Milad Mohareb,Mashari A. Al-Sharif

Research Article

Novel Nicotinonitrile Derivatives Bearing Imino Moieties Enhance Apoptosis and Inhibit Tyrosine Kinase

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 1589-1598
Author(s): Maher A. El-Hashash,Eman A. El-Bordany,Magda I. Marzouk,Abeer M. El-Naggar,Tarek M.S. Nawar,Wael M. El-Sayed

Review Article

Anaplastic Lymphoma Kinase in Glioblastoma: Detection/Diagnostic Methods and Therapeutic Options

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 13 Issue: 2 Year: 2018 Page: 209-223
Author(s): Theodosis Kalamatianos,Despoina Denekou,George Stranjalis,Evangelia Papadimitriou

Review Article

Stemness Phenotype in Tamoxifen Resistant Breast Cancer Cells May be Induced by Interactions Between Receptor Tyrosine Kinases and ER α-66

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 13 Issue: 3 Year: 2018 Page: 302-307
Author(s): Leila Farahmand,Sepideh Mansouri,Narges Jafarbeik-Iravani,Azin Teymourzadeh,Keivan Majidzadeh-A

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