Search Result "morpholine"


Research Article

Synthesis of Imidazo[1,2-b]pyridazine Comprised Piperazine, Morpholine Derivatives as Potent Antimycobacterial Agents with In Vivo Locomotor Activity

Journal: Anti-Infective Agents
Volume: 15 Issue: 2 Year: 2017 Page: 131-139
Author(s): K.R. Paidi,V.B. Tatipamula,M.K. Kolli,S.S.P. Annam,V.R. Pedakotla

Review Article

Balancing Antioxidant, Hypolipidemic and Anti-inflammatory Activity in a Single Agent: The Example of 2-Hydroxy-2-Substituted Morpholine, 1,4-Benzoxazine and 1,4-Benzothiazine Derivatives as a Rational Therapeutic Approach against Atherosclerosis

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 1 Year: 2017 Page: 1214-1227
Author(s): Alexios N. Matralis,Eugenia-Ismini Bavavea,Sandra Incerpi,Jens Z. Pedersen,Angeliki P. Kourounakis

Research Article

A Novel Method for Preparation of Linezolid, (S)-N-((3-(3-Fluoro-4- Morpholinophenyl)-2-Oxo-5-Oxazolidinyl) Methyl) Acetamide

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 1 Year: 2017 Page: 56-60
Author(s): Kondaiah Seku,Vijayakumar Badathala,Venkata Srinivasa Rao Velivela,Srinivasa Reddy Desireddy

Research Article

Synthesis of Mannich Bases by Two Different Methods and Evaluation of their Acetylcholine Esterase and Carbonic Anhydrase Inhibitory Activities

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 5 Year: 2017 Page: 573-580
Author(s): Halise I. Gul,Alkan Demirtas,Gokbay Ucar,Parham Taslimi,Ä°lhami Gulcin

Research Article

Docking-Related Survey on Natural-Product-Based New Monoamine Oxidase Inhibitors and Their Therapeutic Potential

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 6 Year: 2017 Page: 474-491
Author(s): Priyanka Dhiman,Neelam Malik,Anurag Khatkar

Research Article

Novel Mannich-bases as Potential Anticonvulsants: Syntheses, Characterization and Biological Evaluation

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 219-228
Author(s): Amit K. Keshari,Aseem Tewari,Shweta S. Verma,Shailendra K. Saraf

Research Article

Investigation of Ocular Bioactivation Potential and the Role of Cytochrome P450 2D Enzymes in Rat

Journal: Drug Metabolism Letters
Volume: 11 Issue: 2 Year: 2017 Page: 102-110
Author(s): Jennifer L. Dumouchel,Upendra A. Argikar,Jaimie Spear,Ann Brown,Christine E. Dunne,Valerie M. Kramlinger,Amanda L. Cirello,Mithat Gunduz

Research Article

Synthesis and Antiproliferative Activity of New pyrazolo[3,4-c]pyridines

Journal: Medicinal Chemistry
Volume: 13 Issue: 4 Year: 2017 Page: 365-374
Author(s): Efthymios-Spyridon Gavriil, Nikolaos Lougiakis, Nicole Pouli, Panagiotis Marakos, Alexios-Leandros Skaltsounis, Sangkil Nam, Richard Jove, David Horne, Katerina Gioti, Harris Pratsinis, Dimitris Kletsas, Roxane Tenta

Research Article

Synthesis and Study of Analgesic and Anti-inflammatory Activities of Amide Derivatives of Ibuprofen

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 9 Year: 2017 Page: 799-804
Author(s): Abbas Ahmadi, Mohsen Khalili, Zahra Olama, Shirin Karami, Babak Nahri-Niknafs

Research Article

Novel [1,2,4] Triazol [4,3-a] Pyridine Derivatives as Potential Selective c-Met Inhibitors with Improved Pharmacokinetic Properties

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 8 Year: 2017 Page: 1102-1112
Author(s): Junjun Zhao,Shaohua Gou,Xiaobing Zhang,Yan Liang,Lei Fang

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