Search Result "inverse agonists"


Review Article

QSAR Modeling of Histamine H3R Antagonists/inverse Agonists as Future Drugs for Neurodegenerative Diseases

Journal: Current Neuropharmacology
Volume: 16 Issue: 6 Year: 2018 Page: 749-757
Author(s): Michelle Fidelis Correa,Joao Paulo dos Santos Fernandes

Cannabinoid Receptor G Protein-Coupling and Inverse Agonism

Journal: Current Neuropharmacology
Volume: 2 Issue: 1 Year: 2004 Page: 31-36
Author(s): Deborah L. Lewis

Development of New Drugs that Act Through Membrane Receptors and Involve an Action of Inverse Agonism

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 1 Issue: 2 Year: 2006 Page: 207-217
Author(s): Rafael Rodriguez-Puertas, Gabriel Barreda-Gomez

Atypical antipsychotics and inverse agonism at 5-HT2 receptors

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 26 Year: 2015 Page: 3732-3738
Author(s): Laura C. Sullivan,William P Clarke,Kelly A. Berg

Intrinsic Activity at Adenosine A1 Receptors: Partial and Inverse Agonism

Journal: Current Pharmaceutical Design
Volume: 8 Issue: 2 Year: 2002 Page: 2333-2344
Author(s): Rianne A.F. de Ligt, Ad P. Ijzerman

Drugs that Act Through Membrane Receptors and Involve an Action of Inverse Agonism

Ebook: Young People’s Visions of the World

Volume: 1 Year: 2010
Author(s): Gabriel Barreda-Gomez, Rafael Rodriguez-Puertas
Doi: 10.2174/97816080515951100101

Constitutive Activity of Brain Serotonin Receptors: Inverse Agonist Activity of Antipsychotic Drugs

Ebook: Young People’s Visions of the World

Volume: 1 Year: 2010
Author(s): Anil Purohit,Katharine Herrick-Davis,Milt Teitler
Doi: 10.2174/97816080520421040101

Current Knowledge on the Antagonists and Inverse Agonists of Cannabinoid Receptors

Journal: Current Medicinal Chemistry
Volume: 12 Issue: 1 Year: 2005 Page: 1361-1394
Author(s): G. G. Muccioli, D. M. Lambert

Research Article

Discovery and Optimization of a Series of Sulfonamide Inverse Agonists for the Retinoic Acid Receptor-Related Orphan Receptor-α

Journal: Medicinal Chemistry
Volume: 15 Issue: 6 Year: 2019 Page: 674-682
Author(s): Christelle Doebelin,Yuanjun He,Sean Campbell,Philippe Nuhant,Naresh Kumar,Marcel Koenig,Ruben Garcia-Ordonez,Mi Ra Chang,William R. Roush,Li Lin,Susan Kahn,Michael D. Cameron,Patrick R. Griffin,Laura A. Solt,Theodore M. Kamenecka

GABAA Receptor Subtype-Selective Modulators. II. α5-Selective Inverse Agonists for Cognition Enhancement

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 9 Year: 2011 Page: 1203-1214
Author(s): John R. Atack

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