Search Result "enzyme inhibition kinetics"


Research Article

An Investigation of Sodium Fusidate and Recombinant Cytochrome P450 Enzymes Inhibition In-Vitro

Journal: Drug Metabolism Letters
Volume: 10 Issue: 3 Year: 2016 Page: 180-186
Author(s): John Mishriky, Jacqueline Balassone, Zenah Bashour, Simranjit Kaur, Vini Raman, Robel Getachew, Narin Osman, Daniel Guidone, Vincent Chan, Peter J. Little

Binding of Cimetidine to Balb/C Mouse Liver Catalase; Kinetics and Conformational Studies

Journal: Current Clinical Pharmacology
Volume: 11 Issue: 1 Year: 2016 Page: 21-27
Author(s): Mahboubeh Jahangirvand,Dariush Minai-Tehrani,Fatemeh Yazdi,Arash Minai-Tehrani,Nematollah Razmi

Enzymatic and Inhibition Mechanism of Human Aromatase (CYP19A1) Enzyme. A Computational Perspective from QM/MM and Classical Molecular Dynamics Simulations

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 14 Year: 2016 Page: 1112-1124
Author(s): Jacopo Sgrignani,Andrea Cavalli,Giorgio Colombo,Alessandra Magistrato

Calcium Homeostasis and Kinetics in Heart Failure

Journal: Medicinal Chemistry
Volume: 12 Issue: 2 Year: 2016 Page: 151-161
Author(s): Periklis A. Davlouros,Vasileios Gkizas,Chrysoula Vogiatzi,Georgios Giannopoulos,Dimitrios Alexopoulos,Spyridon Deftereos

Research Article

A Novel Liquid Chromatography Tandem Mass Spectrometry Method for the Estimation of Bilirubin Glucuronides and its Application to In Vitro Enzyme Assays

Journal: Drug Metabolism Letters
Volume: 10 Issue: 4 Year: 2016 Page: 264-269
Author(s): Siva P. Putluru,Murali K. Matta,Deepak Ahire,Murali Subramanian,Michael Sinz,Sandhya Mandlekar

Metabolic Enzymes of Helminth Parasites: Potential as Drug Targets

Journal: Current Protein & Peptide Science
Volume: 17 Issue: 3 Year: 2016 Page: 280-295
Author(s): David J. Timson

Review Article

Transformations, Inhibition and Inhibition Control Methods of Sulfur in Sludge Anaerobic Digestion: A Review

Journal: Current Organic Chemistry
Volume: 20 Issue: 2 Year: 2016 Page: 2780-2789
Author(s): Guang Yang, Guangming Zhang, Run Zhuan, Anqi Yang, Yuanyuan Wang

open access plus

Kinetics for Zinc Ion Induced Sepia Pharaonis Arginine Kinase Inactivation and Aggregation

Journal: Protein & Peptide Letters
Volume: 23 Issue: 6 Year: 2016 Page: 508-517
Author(s): Yue-Xiu Si,Jinhyuk Lee,Juan-Ge Cheng,Shang-Jun Yin,Yong-Doo Park,Guo-Ying Qian,Xia-Min Jiang

Flavonoids as Natural Inhibitors of Jack Bean Urease Enzyme

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 3 Year: 2016 Page: 243-249
Author(s): Jalaluddin A. J. Awllia,Maryam AL-Ghamdi,Etimad Huwait,Sumaira Javaid,Atia-tul-Wahab,Saima Rasheed,M. Iqbal Choudhary

Review Article

Expression and Regulation of Drug Transporters and Metabolizing Enzymes in the Human Gastrointestinal Tract

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 39 Year: 2016 Page: 4468-4489
Author(s): M. Drozdzik,S. Oswald

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