Search Result "clogp"


Review Article

Homologation: A Versatile Molecular Modification Strategy to Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 1734-1750
Author(s): Lídia M. Lima,Marina A. Alves,Daniel N. do Amaral

Review Article

Strategically Placed Trifluoromethyl Substituent in the Realm of Antitubercular Drug Design

Journal: Current Drug Therapy
Volume: 14 Issue: 2 Year: 2019 Page: 114-123
Author(s): Sidhartha S. Kar,Cinu A. Thomas

Research Article

Identify Compounds' Target Against Alzheimer's Disease Based on In-Silico Approach

Journal: Current Alzheimer Research
Volume: 16 Issue: 3 Year: 2019 Page: 193-208
Author(s): Yan Hu,Guangya Zhou,Chi Zhang,Mengying Zhang,Qin Chen,Linfeng Zheng,Bing Niu

Research Article

Pyrazole and imidazo[1,2-b]pyrazole Derivatives as New Potential Antituberculosis Agents

Journal: Medicinal Chemistry
Volume: 15 Issue: 1 Year: 2019 Page: 17-27
Author(s): Elda Meta,Chiara Brullo,Michele Tonelli,Scott G. Franzblau,Yuehong Wang,Rui Ma,Wan Baojie,Beatrice S Orena,Maria Rosalia Pasca,Olga Bruno

Research Article

Design, Synthesis and Biological Evaluation of Carbazole Derivatives as Antitubercular and Antibacterial Agents

Journal: Current Bioactive Compounds
Volume: 15 Issue: 1 Year: 2019 Page: 83-97
Author(s): Satheeshkumar Sellamuthu,Mohammad Faizan Bhat,Ashok Kumar,Gopal Nath,Sushil Kumar Singh

Research Article

Synthesis and Investigation on the Antidiabetic Effect of 3-aryl-1-(5-methylisoxazol-3-ylamino)-1-(4-nitrophenyl) Propan-1-one

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 8 Year: 2019 Page: 835-845
Author(s): Jinyu Liu,Zuwen Zhou,Jian Liu,Jufang Yan,Li Fan,Xuemei Tang,Jie Liu,Feifei Chen,Dacheng Yang

Review Article

Identification of Inhibitors against Botulinum Neurotoxins: 8-Hydroxyquinolines Hold Promise

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 1694-1706
Author(s): Ritika Chauhan,Vinita Chauhan,Priyanka Sonkar,Ram Kumar Dhaked

Research Article

Synthesis and Antibacterial Activity of Mefloquine-Based Analogs Against Sensitive and Resistant Mycobacterium tuberculosis Strains

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 9 Year: 2019 Page: 683-689
Author(s): Adriele da Silva Araújo,Adriana M. Moraes,Maria C.S. Lourenço,Cláudia O. Pessoa,Emerson T. da Silva,Marcus V.N. de Souza

Research Article

Vanillin-Related N-Acylhydrazones: Synthesis, Antischistosomal Properties and Target Fishing Studies

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 1241-1251
Author(s): Daniela G.G. Rando,Marcela O.L. da Costa,Thais F.A. Pavani,Thiago Oliveira,Paloma F. dos Santos,Carina R. Amorim,Pedro L.S. Pinto,Mariana G. de Brito,Marcos P.N. Silva,Daniel B. Roquini,Josué de Moraes

Review Article

Fructose-1,6-bisphosphatase Inhibitors: A Review of Recent (2000- 2017) Advances and Structure-Activity Relationship Studies

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 2 Year: 2019 Page: 5542-5563
Author(s): Sarbjit Singh,Dipesh S. Harmalkar,Yongseok Choi,Kyeong Lee

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