Search Result "channel activation and blockade"


Insights into the Molecular Mechanism of hERG1 Channel Activation and Blockade by Drugs

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2010 Page: 3514-3532
Author(s): S. Durdagi, J. Subbotina, J. Lees-Miller, J. Guo, H. J. Duff, S. Y. Noskov

Trafficking of Neuronal Two Pore Domain Potassium Channels

Journal: Current Neuropharmacology
Volume: 8 Issue: 3 Year: 2010 Page: 276-286
Author(s): Alistair Mathie, Kathryn A. Rees, Mickael F. El Hachmane, Emma L. Veale

An Update on Peptide Drugs for Voltage-Gated Calcium Channels

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 5 Issue: 1 Year: 2010 Page: 14-22
Author(s): Lei Gao

Experimental Diabetes Mellitus Down-Regulates Large-Conductance Ca2+- Activated K+ Channels in Cerebral Artery Smooth Muscle and Alters Functional Conductance

Journal: Current Neurovascular Research
Volume: 7 Issue: 2 Year: 2010 Page: 75-84
Author(s): Yan Wang, Hong-Tao Zhang, Xing-Li Su, Xiu-Ling Deng, Bing-Xiang Yuan, Wei Zhang, Xin-Feng Wang, Yu-Bai Yang

TRPC Channels and their Implications for Neurological Diseases

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 9 Issue: 1 Year: 2010 Page: 94-104
Author(s): Senthil Selvaraj, Yuyang Sun, Brij B. Singh

Neurotoxicity of β-Amyloid Protein: Oligomerization, Channel Formation and Calcium Dyshomeostasis

Journal: Current Pharmaceutical Design
Volume: 16 Issue: 2 Year: 2010 Page: 2779-2789
Author(s): Masahiro Kawahara

Endocannabinoids as Regulators of Transient Receptor Potential (TRP)Channels: a Further Opportunity to Develop New Endocannabinoid-Based Therapeutic Drugs

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2010 Page: 1430-1449
Author(s): V. Di Marzo, L. De Petrocellis

Calcium Channel Blockers in Obesity-Related Hypertension

Journal: Immunology, Endocrine & Metabolic Agents in Medicinal Chemistry
Volume: 10 Issue: 2 Year: 2010 Page: 66-75
Author(s): Kazuko Masuo, Gavin W. Lambert

Use of Kv1.3 Blockers for Inflammatory Skin Conditions

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 2 Year: 2010 Page: 2882-2896
Author(s): W. Nguyen, B.L. Howard, D.S. Neale, P.E. Thompson, P.J. White, H. Wulff, D.T. Manallack

The Enigmatic Drug Binding Site for Sodium Channel Inhibitors

Journal: Current Molecular Pharmacology
Volume: 3 Issue: 3 Year: 2010 Page: 129-144
Author(s): Arpad Mike, Peter Lukacs

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