Search Result "admet"


Research Article

In-silico Design, ADMET Screening, MM-GBSA Binding Free Energy of Some Novel Isoxazole Substituted 9-anilinoacridines as HER2 Inhibitors Targeting Breast Cancer

Journal: Current Drug Research Reviews
Volume: 11 Issue: 2 Year: 2019 Page: 118-128
Author(s): Rajagopal Kalirajan,Arumugasamy Pandiselvi,Byran Gowramma,Pandiyan Balachandran

Editorial free to download

Studies of ADMET Properties in Medicinal Chemistry – Part-I

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 2641-2642
Author(s): Luciana Scotti,Marcus Tullius Scotti

Research Article

In-silico Designing, ADMET Analysis, Synthesis and Biological Evaluation of Novel Derivatives of Diosmin Against Urease Protein and Helicobacter pylori Bacterium

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 2658-2675
Author(s): Ritu Kataria,Anurag Khatkar

Research Article

2,4-Dichloro-5-[(N-aryl/alkyl)sulfamoyl]benzoic Acid Derivatives: In Vitro Antidiabetic Activity, Molecular Modeling and In silico ADMET Screening

Journal: Medicinal Chemistry
Volume: 15 Issue: 2 Year: 2019 Page: 186-195
Author(s): Samridhi Thakral,Vikramjeet Singh

Editorial free to download

Studies of ADMET Properties in Medicinal Chemistry – Part-II

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 2742-2742
Author(s): Marcus Tullius Scotti,Luciana Scotti

Research Article

QSAR and Docking Studies on Piperidyl-cyclohexylurea Derivatives for Prediction of Selective and Potent Inhibitor of Matriptase

Journal: Current Computer-Aided Drug Design
Volume: 15 Issue: 2 Year: 2019 Page: 167-181
Author(s): Agha Zeeshan Mirza,Hina Shamshad

General Research Article

Design, Synthesis and In Vitro Evaluation of Novel Anti-HIV 3-Pyrazol-3- yl-Pyridin-2-One Analogs

Journal: Medicinal Chemistry
Volume: 15 Issue: 5 Year: 2019 Page: 561-570
Author(s): Sanjay Kumar,Shiv Gupta,Shraddha Gaikwad,Leila F. Abadi,Late K. K. Bhutani,Smita Kulkarni,Inder P. Singh

Research Article

Search for Potential Inducible Nitric Oxide Synthase Inhibitors with Favorable ADMET Profiles for the Therapy of Helicobacter pylori Infections

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 2795-2804
Author(s): Ricardo Pereira Rodrigues,Juliana Santa Ardisson,Rita de Cássia Ribeiro Gonçalves,Tiago Branquinho Oliveira,Vinicius Barreto da Silva,Daniel Fábio Kawano,Rodrigo Rezende Kitagawa

Research Article

Lead Optimization Studies Towards Finding NS2B/NS3 Protease Targetspecific Inhibitors as Potential Anti-dengue Drug-like Compounds

Journal: Current Drug Discovery Technologies
Volume: 16 Issue: 3 Year: 2019 Page: 307-314
Author(s): Murugaboopathi Gurusamy,Jainul Fathima Abdul

Research Article

Ligand-Based Pharmacophore Modeling and Virtual Screening to Discover Novel CYP1A1 Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 2782-2794
Author(s): Rana Adnan Tahir,Farwa Hassan,Abdul Kareem,Umer Iftikhar,Sheikh Arslan Sehgal

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