Search Result "Thiourea"


Research Article

Synthesis and Biological Activity of Some [(5-oxazolyl)-phenyl]-thiourea Derivatives

Journal: Anti-Infective Agents
Volume: 19 Issue: 1 Year: 2021 Page: 19-27
Author(s): Zhaojin Zhong,Guoling Xing,Jun Liu,Limin Zuo,Zhihui Zheng,Yuhuan Li,Ziwei Huo,Rongmei Gao,Zhuorong Li

Research Article

Synthesis and Erythroid Induction Activity of New Thiourea Derivatives

Journal: Medicinal Chemistry
Volume: 17 Issue: 2 Year: 2021 Page: 121-133
Author(s): Hina Siddiqui,Sarah Shafi,Hamad Ali,Syed Ghulam Musharraf

Research Article

Synthesis of New Thioureas Derivatives and Evaluation of Their Efficacy as Proliferation Inhibitors in MCF-7 Breast Cancer Cells by Using 99mTc-MIBI Radiotracer

Journal: Medicinal Chemistry
Volume: 17 Issue: 7 Year: 2021 Page: 766-778
Author(s): Ahmad Hormati,Jafar Abbasi Shiran,Mikaeil Molazadeh,Babak Kaboudin,Sajjad Ahmadpour

Research Article

Synthesis and Anticancer Activity of Thiadiazole Containing Thiourea, Benzothiazole and Imidazo[2,1-b][1,3,4]thiadiazole Scaffolds

Journal: Medicinal Chemistry
Volume: 17 Issue: 7 Year: 2021 Page: 750-765
Author(s): Stephen Paul Avvaru,Malleshappa N. Noolvi,Uttam A More,Sudipta Chakraborty,Ashutosh Dash,Tejraj M. Aminabhavi,Kumar P. Narayan,Vishnu Sutariya

Research Article

Synthesis and Structure-Activity Relationship Studies of N-monosubstituted Aroylthioureas as Urease Inhibitors

Journal: Medicinal Chemistry
Volume: 17 Issue: 9 Year: 2021 Page: 1046-1059
Author(s): Wei-Wei Ni,Hai-Lian Fang,Ya-Xi Ye,Wei-Yi Li,Li Liu,Zi-Juan Fu,Dawalamu,Wen-Yan Zhu,Ke Li,Fang Li,Xia Zou,Hui Ouyang,Zhu-Ping Xiao,Hai-Liang Zhu

Research Article

Synthesis of Urease Inhibitory 2, 4-bis (4-cyanobenzyl)glycoluril using Sandmeyer Reaction and Density Functional Theory Investigation

Journal: Current Organic Synthesis
Volume: 18 Issue: 0 Year: 2021 Page: 1-6
Author(s): Mirza Arfan Yawer,Shehar Bano,Muhammad Saleem,Affiefa Yawer,Riaz Hussain,Muhammad Imran,Ahmad Irfan,Abdur Rauf,Tareq Abu-Izneid

Research Article

Synthesis and Structure-activity Relationship of Aminoarylthiazole Derivatives as Potential Potentiators of the Chloride Transport Defect in Cystic Fibrosis

Journal: Medicinal Chemistry
Volume: 17 Issue: 6 Year: 2021 Page: 646-657
Author(s): Nara Liessi,Emanuela Pesce,Annalisa Salis,Gianluca Damonte,Bruno Tasso,Elena Cichero,Nicoletta Pedemonte,Enrico Millo

Review Article

Multi-Target Directed Ligands (MTDLs): Promising Coumarin Hybrids for Alzheimer’s Disease

Journal: Current Alzheimer Research
Volume: 18 Issue: 1 Year: 2021 Page: 802-830
Author(s): Rohit Bhatia,Sankha S. Chakrabarti,Upinder Kaur,Gaurav Parashar,Anindita Banerjee,Ravindra K. Rawal

Research Article

Design, Synthesis, Pharmacological evaluation, in silico modeling, prediction of toxicity and metabolism studies of novel 1-(substituted)-2-methyl-3-(4-oxo-2-phenyl quinazolin-3(4H)-yl)isothioureas

Journal: Medicinal Chemistry
Volume: 17 Issue: 4 Year: 2021 Page: 352-368
Author(s): M.T. Sulthana,V. Alagarsamy,K. Chitra

Review Article

Greener Approaches to Selected Asymmetric Addition Reactions Relevant to Drug Development

Journal: Current Organic Chemistry
Volume: 25 Issue: 1 Year: 2021 Page: 1497-1522
Author(s): Girija S. Singh

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