Search Result "Pyrazole."


Discovery and Development of Pyrazole-Scaffold Hsp90 Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 6 Issue: 1 Year: 2006 Page: 1193-1203
Author(s): Edward McDonald, Keith Jones, Paul A. Brough, Martin J. Drysdale, Paul Workman

Synthesis, Biological Evaluation and 3D-QSAR of 1,3,5-Trisubstituted-4,5- Dihydro-(1H)-Pyrazole Derivatives as Potent and Highly Selective Monoamine Oxidase A Inhibitors

Journal: Current Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2006 Page: 1411-1428
Author(s): Franco Chimenti, Adriana Bolasco, Fedele Manna, Daniela Secci, Paola Chimenti, Arianna Granese, Olivia Befani, Paola Turini, Roberto Cirilli, Francesco La Torre, Stefano Alcaro, Francesco Ortuso, Thierry Langer

Convenient Synthesis of Some New Substituted Pyrazolyl-1,3,4-Oxadiazoles and Pyrazolyl-1,2,4- Triazoles

Journal: Letters in Organic Chemistry
Volume: 3 Issue: 3 Year: 2006 Page: 195-200
Author(s): Ahmad M. Farag, Yehya M. Elkholy, Korany A. Ali

Synthesis of Tricyclic Pyrazolo[1,5-a]pyrimidin-7(4H)-ones Featuring Regioselective Formation of the Core Structure

Journal: Letters in Organic Chemistry
Volume: 3 Issue: 9 Year: 2006 Page: 715-719
Author(s): Vladislav Z. Parchinsky, Olga Ushakov, Dmitry V. Kravchenko, Mikhail Krasavin

Highlights in Organic Chemistry [Oxidative Aromatization Using Molecular Oxygen Promoted by Activated Carbon]

Journal: Letters in Organic Chemistry
Volume: 3 Issue: 8 Year: 2006 Page: 571-578
Author(s): Masahiko Hayashi, Yuka Kawashita

Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidine Template: Organic and Medicinal Chemistry Approach

Journal: Current Organic Chemistry
Volume: 10 Issue: 3 Year: 2006 Page: 259-275
Author(s): Hussein El-Kashef, Romeo Romagnoli, Pier G. Baraldi, Mojgan A. Tabrizi, Pier A. Borea, Marina Gordaliza, Delia Preti, Andrea Bovero, Francesca Fruttarolo

Effectiveness of Hsp90 Inhibitors as Anti-Cancer Drugs

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 6 Issue: 1 Year: 2006 Page: 1137-1143
Author(s): Li Xiao, Xiangyi Lu, Douglas M. Ruden

Microwave-Assisted Regiospecific Synthesis of 2-Trifluoromethyl-7- Trihalomethylated Pyrazolo[1,5-a]Pyrimidines

Journal: Letters in Organic Chemistry
Volume: 3 Issue: 5 Year: 2006 Page: 358-362
Author(s): Fernanda A. Rosa, Helio G. Bonacorso, Nilo Zanatta, Alex F.C. Flores, Gabriela F. Fiss, Daniel J. Emmerich, Elisandra Scapin, Marcos A.P. Martins, Wilson Cunico

Anti-Obesity

Journal: Current Bioactive Compounds
Volume: 2 Issue: 1 Year: 2006 Page: 126-126
Author(s): Bentham Science Publisher

Editorial [ Molecular Chaperones as Targets in Medicinal Chemistry and Drug Discovery Guest Editor: Dr. Gabriela Chiosis ]

Journal: Current Topics in Medicinal Chemistry
Volume: 6 Issue: 1 Year: 2006 Page: 1161-1161
Author(s): Gabriela Chiosis

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