Search Result "MDR-inhibitors"


Three Decades of P-gp Inhibitors: Skimming Through Several Generations and Scaffolds

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 13 Year: 2012 Page: 1946-2025
Author(s): A. Palmeira,E. Sousa,M. H. Vasconcelos,M. M. Pinto

Colon Adenocarcinoma Multidrug Resistance Reverted by Euphorbia Diterpenes: Structure-Activity Relationships and Pharmacophore Modeling

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 12 Issue: 9 Year: 2012 Page: 1015-1024
Author(s): Mariana Reis,Ricardo J. Ferreira,Julianna Serly,Noelia Duarte,Ana M. Madureira,Daniel J. V. A. Santos,Joseph Molnar,Maria-Jose U. Ferreira

Cationic Lipophilic Radiotracers for Functional Imaging of Multidrug Resistance

Journal: Current Radiopharmaceuticals
Volume: 5 Issue: 2 Year: 2012 Page: 113-123
Author(s): Celia M.F. Gomes

Structure and Ligand-based Design of P-glycoprotein Inhibitors: A Historical Perspective

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 27 Year: 2012 Page: 4197-4214
Author(s): Andreia Palmeira,Emilia Sousa,M. Helena Vasconcelos,Madalena Pinto,Miguel X. Fernandes

Genomics and Cancer Drug Resistance

Journal: Current Pharmaceutical Biotechnology
Volume: 13 Issue: 5 Year: 2012 Page: 651-673
Author(s): Antonio S. Rodrigues, Joana Dinis, Marta Gromicho, Celia Martins, Antonio Laires, Jose Rueff

The Impact of the Induction of Multidrug Resistance Transporters in Therapies by Used Drugs: Recent Studies

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 11 Year: 2012 Page: 1127-1134
Author(s): A. Hilgeroth,M. Hemmer,C. Coburger

Synthesis and Biological Evaluation of a Series of 6,7-dimethoxy-1-(3,4- dimethoxybenzyl)-2-substituted Tetrahydroisoquinoline Derivatives

Journal: Medicinal Chemistry
Volume: 8 Issue: 4 Year: 2012 Page: 711-716
Author(s): Zhi-hong Zou,Xiao-bu Lan,Chun-lei Tang,Xiao-yun Zhu,Bao-min Liu,Hai Qian,Wen-long Huang,Yun-man Li

UDP-3-O-(R-3-hydroxymyristoyl)-N-Acetylglucosamine Deacetylase (LpxC) Inhibitors: A New Class of Antibacterial Agents

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 13 Year: 2012 Page: 2038-2050
Author(s): J. Zhang,L. Zhang,X. Li,W. Xu

1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story So Far And Perspectives (Part 2): Action in Other Targets and Antitargets

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 25 Year: 2012 Page: 4306-4323
Author(s): E. Carosati,P. Ioan,M. Micucci,F. Broccatelli,G. Cruciani,B.S. Zhorov,A. Chiarini,R. Budriesi

Adenylating Enzymes in Mycobacterium tuberculosis as Drug Targets

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 7 Year: 2012 Page: 766-796
Author(s): Benjamin P. Duckworth,Kathryn M. Nelson,Courtney C. Aldrich

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