Search Result "CYP isoenzymes"


Cunninghamella Biotransformation - Similarities to Human Drug Metabolism and Its Relevance for the Drug Discovery Process

Journal: Current Drug Metabolism
Volume: 17 Issue: 2 Year: 2016 Page: 107-117
Author(s): Kamil Piska, Dorota ?elaszczyk, Marek Jamrozik, Paulina Kubowicz-Kwa?ny, El?bieta P?kala

Research Article

An Investigation of Sodium Fusidate and Recombinant Cytochrome P450 Enzymes Inhibition In-Vitro

Journal: Drug Metabolism Letters
Volume: 10 Issue: 3 Year: 2016 Page: 180-186
Author(s): John Mishriky, Jacqueline Balassone, Zenah Bashour, Simranjit Kaur, Vini Raman, Robel Getachew, Narin Osman, Daniel Guidone, Vincent Chan, Peter J. Little

Insights into the Structural Features Essential for JAK2 Inhibition and Selectivity

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 13 Year: 2016 Page: 1331-1355
Author(s): Chao Zhao,Daulat Bikram Khadka,Won-Jea Cho

In Vitro CYP2D Inhibitory Effect and Influence on Pharmacokinetics and Pharmacodynamic Parameters of Metoprolol Succinate by Terminalia arjuna in Rats

Journal: Drug Metabolism Letters
Volume: 10 Issue: 2 Year: 2016 Page: 124-135
Author(s): Alice Varghese, Jay Savai, Shruti Mistry, Preeti Khandare, Kalyani Barve, Nancy Pandita, Ram Gaud

Pharmacotherapy for Patent Ductus Arteriosus: Current Options and Outstanding Questions

Journal: Current Pediatric Reviews
Volume: 12 Issue: 2 Year: 2016 Page: 110-119
Author(s): Sara E. Rostas,Christopher C. McPherson

Prediction of Metabolism of Drugs using Artificial Intelligence: How far have we reached?

Journal: Current Drug Metabolism
Volume: 17 Issue: 2 Year: 2016 Page: 129-141
Author(s): Rajnish Kumar, Anju Sharma, Mohammed Haris Siddiqui, Rajesh Kumar Tiwari

Research Article

Clopidogrel High On-Treatment Platelet Reactivity in Patients with Carotid Artery Stenosis Undergoing Endarterectomy. A Pilot Study

Journal: Current Vascular Pharmacology
Volume: 14 Issue: 6 Year: 2016 Page: 563-569
Author(s): Dragana Backovic, Svetlana Ignjatovic, Ljiljana Rakicevic, Mirjana Novkovic, Jelena Kusic-Tisma, Dragica Radojkovic, Evgenija Strugarevic, Branko Calija, Djordje Radak, Mirjana Kovac

Influence of CYP3A5 Polymorphism on the Pharmacokinetics of Psychiatric Drugs

Journal: Current Drug Metabolism
Volume: 17 Issue: 3 Year: 2016 Page: 227-236
Author(s): Georgia Ragia, Marja-Liisa Dahl, Vangelis G. Manolopoulos

Mechanisms of Resistance to Chemotherapy in Gastric Cancer

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2016 Page: 318-334
Author(s): J.J.G. Marin,R. Al-Abdulla,E. Lozano,O. Briz,L. Bujanda,J. M. Banales,R.I.R. Macias

Research Article

New Dehydroepiandrosterone-triazole Derivatives Identified as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Enzyme in the Prostate

Journal: Current Enzyme Inhibition
Volume: 12 Issue: 2 Year: 2016 Page: 145-154
Author(s):

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