Search Result "COX"


Review Article

Update on COX-2 Selective Inhibitors: Chemical Classification, Side Effects and their Use in Cancers and Neuronal Diseases

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 26 Year: 2017 Page: 2935-2956
Author(s): Anita-Marie Rayar,Nathalie Lagarde,Clotilde Ferroud,Jean-Francois Zagury,Matthieu Montes,Maite Sylla-Iyarreta Veitia

Research Article

Aryl/heteroaryl Substituted Celecoxib Derivatives as COX-2 Inhibitors: Synthesis, Anti-inflammatory Activity and Molecular Docking Studies

Journal: Medicinal Chemistry
Volume: 13 Issue: 5 Year: 2017 Page: 484-497
Author(s): Golla Madhava,Katla V. Ramana,Saddala M. Sudhana,Devineni S. Rao,Kuntrapakam H. Kumar,Valluru Lokanatha,Asupatri U. Rani,Chamarthi N. Raju

Research Article

Novel Thiourea Derivatives Bearing Sulfonamide Moiety as Anticancer Agents Through COX-2 Inhibition

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 10 Year: 2017 Page: 1411-1425
Author(s): Mostafa M. Ghorab,Mohamed S.A. El-Gaby,Mansour S. Alsaid,Yaseen A.M.M. Elshaier,Aiten M. Soliman,Fardous F. El-Senduny,Farid A. Badria,Abdelrahman Y.A. Sherif

Review Article

A Rat Model of Ischemic Enteritis: Pathogenic Importance of Enterobacteria, iNOS/NO, and COX-2/PGE2

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 27 Year: 2017 Page: 4048-4056
Author(s): Koji Takeuchi,Yoshino Komatsu,Yuka Nakamori,Tohru Kotani

Research Article

Anti-Inflammatory Activity of Novel 12-N-methylcytisine Derivatives

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2017 Page: 112-122
Author(s): Inna P. Tsypysheva,Sophia S. Borisevich,Liana F. Zainullina,Nina S. Makara,Alena V. Koval`skaya,Polina R. Petrova,Sergey L. Khursan,Yulia V. Vakhitova,Felix S. Zarudii

Review Article

Cardiovascular Toxicity of Cyclooxygenase Inhibitors and Promising Natur a l Substitutes

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 6 Year: 2017 Page: 952-960
Author(s): Mahmoud Bahmani,Amir Sarrafchi,Hedayatollah Shirzad,Sedigheh Asgari,Mahmoud Rafieian-Kopaei

Research Article

In vitro and In silico: Selectivities of Seychellene Compound as Candidate Cyclooxygenase Isoenzyme Inhibitor on Pre-Osteoblast Cells

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 1 Year: 2017 Page: 2-10
Author(s): Sentot J. Raharjo,Chanif Mahdi,Nurdiana Nurdiana,Takheshi Kikuchi,Fatchiyah Fatchiyah

Research Article

Molecular Docking and Structure Activity Relationship Studies of NSAIDs. What do they Reveal about IC50?

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 8 Year: 2017 Page: 949-958
Author(s): Chrysoula Mikra,Georgios Rossos,Sotirios K. Hadjikakou,Nikolaos Kourkoumelis

Research Article

Synthesis of New Thiazolyl Coupled Pyrazoles Bearing 2,4-Thiazolidinedionyl Pharmacophore and Their Anti-Inflammatory and Antibacterial Evaluation

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2017 Page: 46-57
Author(s): Lalit Khillare,Manisha Bhosle,Mahendra Bhalerao,Kiran Kharat,Ramrao Mane

Research Article

A Purified Fraction of Ocimum tenuiflorum (L) Inhibits LTC4, LTA4 and COX-2 Activities, Down-Regulates mRNA Expression in HL-60 Cells and Reduces Lung Inflammation in an OVA Induced Asthma Model in BALB/c Mice

Journal: Immunology, Endocrine & Metabolic Agents in Medicinal Chemistry (Discontinued)
Volume: 17 Issue: 2 Year: 2017 Page: 115-126
Author(s): Kapil K. Soni,Nishikant Raut,Temitope O. Lawal,Udeshi Patel,Gail B. Mahady

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