Search Result "COMFA"


Research Article

In Silico ADME and QSAR Studies on a Set of Coumarin Derivatives As Acetylcholinesterase Inhibitors Against Alzheimer’s Disease: CoMFA, CoMSIA, Topomer CoMFA, and HQSAR

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 6 Year: 2020 Page: 684-712
Author(s): Uttam A. More,Sameera Patel,Vidhi Rahevar,Malleshappa N. Noolvi,Tejraj M. Aminabhavi,Shrinivas D. Joshi

Research Article

Molecular modelling studies on thiazole-based α-Glucosidase Inhibitor using docking and CoMFA, CoMSIA and HQSAR

Journal: Current Drug Discovery Technologies
Volume: 17 Issue: 0 Year: 2020 Page: 1-19
Author(s): Deshbandhu Joshi,Shourya Yadav,Rajesh Sharma,Mitrunjaya Pandya,Raghvendra Singh Bhadauria

Research Article

QSAR Studies of Sulfonamide Hydroxamates Derivatives as MMP-2 Inhibitors Topomer CoMFA and Molecular Docking

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 1 Year: 2020 Page: 1364-1371
Author(s): Jian-Bo Tong,Feng Yi,Ding Luo,Tian-Hao Wang

Research Article

CoMFA, CoMSIA and HQSAR Analysis of 3-aryl-3-ethoxypropanoic Acid Derivatives as GPR40 Modulators

Journal: Current Drug Discovery Technologies
Volume: 17 Issue: 1 Year: 2020 Page: 100-118
Author(s): Krishna A. Gajjar,Anuradha K. Gajjar

Research Article

Molecular Modeling Studies of Anti-Alzheimer Agents by QSAR, Molecular Docking and Molecular Dynamics Simulations Techniques

Journal: Medicinal Chemistry
Volume: 16 Issue: 7 Year: 2020 Page: 903-927
Author(s): Rahman Abdizadeh,Farzin Hadizadeh,Tooba Abdizadeh

Research Article

Novel 1,2,3-Triazole-functionalized pyrido[3',2':4,5]furo[3,2-d]pyrimidin- 4(3H)-one Derivatives: Synthesis, Anticancer Activity, CoMFA and CoMSIA Studies

Journal: Letters in Organic Chemistry
Volume: 17 Issue: 1 Year: 2020 Page: 969-978
Author(s): Sailu Betala,Balakishan Vadla

Research Article

Three-dimensional Quantitative Structure-activity Relationship (3DQSAR) and Molecular Docking Study of 2-((pyridin-3-yloxy)methyl) Piperazines as α7 Nicotinic Acetylcholine Receptor Modulators for the Treatment of Inflammatory Disorders

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1031-1041
Author(s): Deepika Purohit,Vandana Saini,Sanjiv Kumar,Ajit Kumar,Balasubramanian Narasimhan

Research Article

3D-QSAR and Docking Studies on Pyrimidine Derivatives as CSF-1R inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 3 Year: 2020 Page: 341-355
Author(s): Ya-ting Deng,Jun-wei Wang,Han Chu,Juan Wang,Yong Hu,Yong lin,Mao Shu,Zhi-hua Lin

Research Article

Integrated Protocol to Design Potential Inhibitors of Dipeptidyl Peptidase- 4 (DPP-4)

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 3 Year: 2020 Page: 209-226
Author(s): Simone Queiroz Pantaleão,Eric Allison Philot,Michell de Oliveira Almeida,Angelica Nakagawa Lima,Mirela Inês de Sairre,Ana Ligia Scott,Kathia Maria Honorio

Research Article

Design of New Therapeutic Agents Targeting FLT3 Receptor Tyrosine Kinase Using Molecular Docking and 3D-QSAR Approach

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 5 Year: 2020 Page: 583-594
Author(s): Swapnil P. Bhujbal,Seketoulie Keretsu,Seung Joo Cho

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