Search Result "Blockade"


Research Article

Targeted Blockade of TARP-γ8-Associated AMPA Receptors: Anticonvulsant Activity with the Selective Antagonist LY3130481 (CERC-611)

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 16 Issue: 1 Year: 2017 Page: 1099-1110
Author(s): Jeffrey M. Witkin,Douglas A. Schober,Scott D. Gleason,John T. Catlow,Warren J. Porter,Jon Reel,Xiaoming Jin,Jonathan Hobbs,Donald Gehlert,Douglas L. Gernert,Kevin M. Gardinier,Akihiko S. Kato,Xingjie Ping,Jodi L. Smith

Research Article

Development of a Radiolabeled Amlodipine Analog for L-type Calcium Channel Imaging

Journal: Current Radiopharmaceuticals
Volume: 10 Issue: 1 Year: 2017 Page: 51-58
Author(s): Tahereh Firouzyar,Amir Reza Jalilian,Mohammad Reza Aboudzadeh,Hossein Sadeghpour,Mehrban Pooladi,Mahdi Shafiee-Ardestani,Ali Khalaj

Research Article

Strong Quantum Confinement Effects in Nanometer Devices with Graphene Directly Grown on Insulator by Catalyst-free Chemical Vapor Deposition

Journal: Current Graphene Science (Discontinued)
Volume: 1 Issue: 1 Year: 2017 Page: 44-48
Author(s): Hiroto Sato,Atsushi Nakamura,Amit Banerjee,Kenji Yamada,Hiroaki Satoh,Jiro Temmyo,Hiroshi Inokawa

Review Article

Inflammatory Bowel Disease: New Therapeutic Options in the Post Anti-TNFα Era

Journal: Current Drug Metabolism
Volume: 18 Issue: 7 Year: 2017 Page: 666-679
Author(s): Miguel Jiménez-Pérez,Raúl V Olmedo-Martín,Víctor M Amo-Trillo,Rocío González-Gande

Review Article

Recent Developments on Multi-Target-Directed Tacrines for Alzheimer's Disease. I. The Pyranotacrines

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 3328-3335
Author(s): Alejandro Romero,Jose Marco-Contelles

Research Article

Diosmetin Induces Cell Apoptosis by Regulating CYP1A1/CYP1A2 Due to p53 Activation in HepG2 Cells

Journal: Protein & Peptide Letters
Volume: 24 Issue: 5 Year: 2017 Page: 406-412
Author(s): Bin Liu,Kaiqiao Jia,Yu Yang,Siyuan Hao,Caijie Lu,Fengming Xu,Dehui Feng,Runzhi Zhu

Research Article

Pharmacological Effects of Turmeric on Learning, Memory and Expression of Muscarinic Receptor Genes (M1, M3 and M5) in Stress-induced Mouse Model

Journal: Current Drug Targets
Volume: 18 Issue: 13 Year: 2017 Page: 1545-1557
Author(s): Aliya Khalid,Rabia Shakeel,Saira Justin,Ghazala Iqbal,Syed Adnan Ali Shah,Saadia Zahid,Touqeer Ahmed

Research Article

Beta-Blockers are Associated with Decreased In-Hospital Mortality and Stroke in Acute Decompensated Heart Failure: Findings from a Retrospective Analysis of a 22-Year Registry in the Middle East (1991-2013)

Journal: Current Vascular Pharmacology
Volume: 15 Issue: 1 Year: 2017 Page: 77-83
Author(s): Charbel Abi Khalil,Jassim Al Suwaidi,Rajvir Singh,Nidal Asaad,Galal Abushahba,Unus Kunju,Awad Al-Qahtani,Hajar A. AlBinali

Review Article

Immunomodulatory Drugs: Immune Checkpoint Agents in Acute Leukemia

Journal: Current Drug Targets
Volume: 18 Issue: 3 Year: 2017 Page: 315-331
Author(s): Hanna A. Knaus,Christopher G. Kanakry,Leo Luznik,Ivana Gojo

Review Article

Emerging Family of Protein-protein Interaction Inhibitors Targeting PD-1 Checkpoint Pathway

Journal: Current Cancer Therapy Reviews
Volume: 13 Issue: 2 Year: 2017 Page: 120-128
Author(s): Yijun Huang,Hong Zhang

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