Search Result "Antagonist"


Research Article

Design, Synthesis, and Evaluation of Isoquinoline Ureas as TRPV1 Antagonists

Journal: Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2020 Page: 202-211
Author(s): Nehaben A. Gujarati,Bradley J. Undem,Vijaya L. Korlipara

General Review Article

Aldosterone and Mineralocorticoid Receptor Antagonists on Pulmonary Hypertension and Right Ventricular Failure: A Review

Journal: Current Pharmaceutical Design
Volume: 26 Issue: 3 Year: 2020 Page: 3862-3870
Author(s): Navid Omidkhoda,Farveh Vakilian,Amir Hooshang Mohammadpour,Thozhukat Sathyapalan,Amirhossein Sahebkar

Mini-Review Article

Factors Affecting the Wear Behavior of Monolithic Zirconia and the Antagonists: Literature Review

Journal: Current Dentistry
Volume: 2 Issue: 1 Year: 2020 Page: 4-11
Author(s): Marcia Borba,Paula Benetti,Giordana P. Furini,Kátia R. Weber,Tábata M. da Silva

Research Article

Design, Synthesis and Evaluation of Novel Substituted (5-methyl-1H-pyrazol-3-yl)- 1,3,4-oxadiazole as Potent Androgen Receptor Antagonist

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 84-93
Author(s): Sasikumar Andavar,Mohanasrinivasan Vaithilingam,Divakar Selvaraj,Ajeeshkumar A. Kumaran,Krishnaswamy Devanathan

Systematic Review Article

Non-Vitamin K Antagonist Oral Anticoagulants in Pulmonary Embolism: An Overview of Systematic Reviews

Journal: Current Pharmaceutical Design
Volume: 26 Issue: 2 Year: 2020 Page: 2686-2691
Author(s): Ioannis Doundoulakis,Christina Antza,Haralambos Karvounis,George Giannakoulas

Review Article

Triple Negative Breast Cancer: How Neurokinin-1 Receptor Antagonists Could Be Used as a New Therapeutic Approach

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 20 Issue: 5 Year: 2020 Page: 408-417
Author(s): Miguel Muñoz,Marisa Rosso,Rafael Coveñas

Review Article

Radiolabeled GRPR Antagonists for Imaging of Disseminated Prostate Cancer. Influence of Labeling Chemistry on Targeting Properties

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 4 Year: 2020 Page: 7090-7111
Author(s): Bogdan Mitran,Vladimir Tolmachev,Anna Orlova

Research Article

Relationship Between Polymorphisms of Interleukin-1 Receptor Antagonist (IL-1Ra) Genes and Susceptibility to Systemic Lupus Erythematosus in Iranian Population

Journal: Current Rheumatology Reviews
Volume: 16 Issue: 2 Year: 2020 Page: 84-88
Author(s): Rashin Ganjali,Jalil Tavakkol Afshari,Zahra Rezaieyazdi,Mandana Khodashahi,Azam Brook,Maryam Mazhani,Mohamad Reza Hatef,Mahnaz Abbasi

Research Article open access plus

Preparation and Evaluation of Polymeric Microparticles of Human Recombinant IL-1 Receptor Antagonist by Spray Drying

Journal: Drug Delivery Letters
Volume: 10 Issue: 4 Year: 2020 Page: 308-313
Author(s): Anand Ubhe,Gerard G.M. D’Souza

Research Article

Studies on the IC50 of Metabolically Stable 1-(3,3-diphenylpropyl)- piperidinyl Amides and Ureas as Human CCR5 Receptor Antagonists Based on QSAR

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 8 Year: 2020 Page: 1036-1046
Author(s): Yutao Zhao,Xiaoqian Liu,Jing Ouyang,Yan Wang,Shanyu Xu,Dongdong Tian,Hongzong Si

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