Search Result "ADME evaluation ."


Synthesis and Preliminary Biological Evaluation of Polyamine-aniline Acridines as P-glycoprotein Inhibitors

Journal: Medicinal Chemistry
Volume: 10 Issue: 5 Year: 2014 Page: 506-511
Author(s): Jianhong Wang,Pengfei Cheng,Tianwei Luo,Zhaoyi Wang,Yahong Zhang,Jin Zhao

Evaluation of Herbal Medicines: Value Addition to Traditional Medicines Through Metabolism, Pharmacokinetic and Safety Studies

Journal: Current Drug Metabolism
Volume: 15 Issue: 10 Year: 2014 Page: 942-952
Author(s): Roslyn Thelingwani,Collen Masimirembwa

A Proposed Screening Paradigm for Discovery of Covalent Inhibitor Drugs

Journal: Drug Metabolism Letters
Volume: 8 Issue: 1 Year: 2014 Page: 19-30
Author(s): Mehran F. Moghaddam,Yang Tang,Zhihong O’Brien,Samantha J. Richardson,Maria Bacolod,Prasoon Chaturedi,Julius Apuy,Ashutosh Kulkarni

Molecular Dynamics, Density Functional Theory, Pharmacophore Modeling, Molecular Interaction Fields and ADME/Tox Investigation of Novel Bioactive Compounds Interacting with CDK2 Surfaces

Journal: Current Physical Chemistry
Volume: 4 Issue: 1 Year: 2014 Page: 94-105
Author(s): Fernanda P. Ferreira,Wagner F. Couto,Vanessa Fontana,Carlton A. Taft,Carlos H.T.P. Da Silva

Synthesis and Biological Evaluation of Sulfonilamidothienopyrimidinone Derivatives as Novel Anti-inflammatory Agents

Journal: Medicinal Chemistry
Volume: 10 Issue: 7 Year: 2014 Page: 700-710
Author(s): Mariarita Barone, Andrea Santagati, Adriana C.E. Graziano, Cosimo G. Fortuna, Giuseppe Ronsisvalle, Venera Cardile

Design Potential Selective Inhibitors for Treating Cancer by Targeting the Src Homology 2 (SH2) Domain-Containing Phosphatase 2 (Shp2) with Core Hopping Approach

Journal: Protein & Peptide Letters
Volume: 21 Issue: 6 Year: 2014 Page: 556-563
Author(s): Yu-Qing Duan,Ying Ma,Xue-Jiao Wang,Yuan-Yuan Jin,Run-Ling Wang,Wei-Li Dong,Wei-Ren Xu,De-Xin Kong,Shu-Qing Wang

Virtual Screening Against M. tuberculosis 7,8-Diaminopelargonic Acid Synthase (MtbBioA) and In Silico Toxicity Evaluation of Top Hits

Journal: Current Enzyme Inhibition
Volume: 10 Issue: 2 Year: 2014 Page: 105-112
Author(s): Junie Billones,Maria C. Carrillo,Voltaire Organo,Stephani J. Macalino,Inno Emnacen,Jamie B. Sy

Virtual Screening and Molecular Descriptor Analysis on Dietary Phytochemicals Against Heat Shock Protein 90 Enzyme

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 1 Year: 2014 Page: 40-49
Author(s): Salam Pradeep Singh,Bolin Kumar Konwar

The Survey of the Use of QSAR Methods to Determine Intestinal Absorption and Oral Bioavailability During Drug Design

Journal: Medicinal Chemistry
Volume: 10 Issue: 5 Year: 2014 Page: 441-448
Author(s): Fredson Torres Silva,Gustavo H.G. Trossini

Chitosan Surface-Modified PLGA Nanoparticles: Preparation, Characterization, and Evaluation of their In Vitro Drug-Release Behaviors and Cytotoxicities

Journal: Current Nanoscience
Volume: 10 Issue: 2 Year: 2014 Page: 255-262
Author(s): Hong-li Chen, Yong-xue Wang, Ping Zhou, Rui Liu, Wen-bin Nan, Yin-song Wang, Yong-tao Liu, Yan Wang, Qing-qing Xiong, Hui-gen Feng, Qi-qing Zhang

Previous   Next

Go To   Results 1 - 1 of 81

Filter Result

Volume Year
Content Type
Ads
© 2024 Bentham Science Publishers | Privacy Policy