Search Result "5-1H-1"


An Efficient Synthesis and Antiviral Activity Evaluation of 1-[4-(5-Phenyl- 4, 5 dihydro-1H-pyrazole [& (4, 5 dihydroisoxazole)]-3-yl)-phenyl]-pyrrole- 2, 5-dione Derivates

Journal: Anti-Infective Agents
Volume: 12 Issue: 1 Year: 2014 Page: 104-111
Author(s): Jigarkumar Patel,Mahesh Malani,Graciela Andrei,Jan Balzarini,Robert Snoeck,Bharat Dholakiya

Synthesis, Pharmacological Activity and Molecular Modeling of 1-Aryl-7- hydroxy-2,3-dihydroimidazo[1,2-a]pyrimidine-5(1H)-ones and their 6-Substituted Derivatives

Journal: Medicinal Chemistry
Volume: 10 Issue: 5 Year: 2014 Page: 460-475
Author(s): Marzena Rzadkowska,Elzbieta Szacon,Agnieszka A. Kaczor,Sylwia Fidecka,Ewa Kedzierska,Dariusz Matosiuk

Synthesis, Characterization and Antitumor Activity of Novel Triazole/ Isoxazole Tagged Pyridine Hybrids

Journal: Letters in Organic Chemistry
Volume: 11 Issue: 4 Year: 2014 Page: 293-302
Author(s): Raju K, Chandra Shekhar A, Sathaiah G, Ravi Kumar A, Narsaiah B, Shanthan Rao P, Srujana R, Srigiridhar Kotamraju

Synthesis and Evaluation of N-Substituted Thiazolidine-2,4-dione Containing Pyrazole as a Potent Antimicrobial Agents

Journal: Anti-Infective Agents
Volume: 12 Issue: 1 Year: 2014 Page: 85-94
Author(s): Nisheet C. Desai,Hitesh M. Satodiya,Kiran M. Rajpara,Vivek V. Joshi,Kandarp Bhatt,Hasit V. Vaghani

Synthesis and Dual D2 and 5-HT1A Receptor Binding Affinities of 7-piperazinyl and 7-piperidinyl-3,4-dihydroquinazolin-2(1H)-ones

Journal: Medicinal Chemistry
Volume: 10 Issue: 5 Year: 2014 Page: 484-496
Author(s): Nisar Ullah

Structural Studies on N-(1-naphthyl)-3-amino-5-oxo-4-phenyl-1Hpyrazole- 1-carboxamide with Antibacterial Activity

Journal: Letters in Organic Chemistry
Volume: 11 Issue: 1 Year: 2014 Page: 40-48
Author(s): Agnieszka A. Kaczor, Tomasz Wrobel, Zbigniew Karczmarzyk, Waldemar Wysocki, Andrzej Fruzinski, Malgorzata Brodacka, Dariusz Matosiuk, Monika Pitucha

Positive Allosteric Modulators (PAMs) of Metabotropic Glutamate Receptor 5 (mGluR5) Attenuate Microglial Activation

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 13 Issue: 4 Year: 2014 Page: 558-566
Author(s): Fengtian Xue,Bogdan A. Stoica,Marie Hanscom,Shruti V. Kabadi,Alan I. Faden

Novel 4-bromo-2-(3-methyl-1-(substituted-phenylsulfonyl)-4,5-dihydro-1- H-pyrazol-5-yl)phenol Derivatives: Synthesis and Antibacterial Activity

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 5 Year: 2014 Page: 572-577
Author(s): Qing Chenga, Ying-Ming Jia, Fei-Hu Cheng, Xin-Hua Liu

Cu-mediated synthesis of 2,3-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-1-ones as potential inhibitors of sirtuins

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 2 Year: 2014 Page: 199-206
Author(s): Sreerama Srinivas Rao,Dandela Rambabu,Mohosin Layek,Kummari Lalith Kumar,Mandava Venkata Basaveswara Rao,Devyani Haldar,Manojit Pal

Evaluation of Structural Effects of Acyclic and Macrocyclic Ligands Derived from (R,R)-Cyclohexane-1,2-diamine in the Enantioselective Cu(II)-Catalyzed Henry Reaction

Journal: Letters in Organic Chemistry
Volume: 11 Issue: 9 Year: 2014 Page: 633-638
Author(s): Lucia Cerisoli,Stefano Grilli,Diego Savoia

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