Search Result "4- thiadiazole"


Research Article

Design, Synthesis, Molecular Docking and In silico Analysis of Some Novel 2-Amino-1, 3, 4-Thiadiazole Derivatives as Potent DNA Gyrase B Inhibitors

Journal: Current Bioactive Compounds
Volume: 17 Issue: 7 Year: 2021 Page: 8-17
Author(s): Natarajan Ramalakshmi,Prabakaran A.,Sumithra S.,Keerthika S.,Nivetha J.,Raveena R.

Research Article

Synthesis and Anticancer Activity of Thiadiazole Containing Thiourea, Benzothiazole and Imidazo[2,1-b][1,3,4]thiadiazole Scaffolds

Journal: Medicinal Chemistry
Volume: 17 Issue: 7 Year: 2021 Page: 750-765
Author(s): Stephen Paul Avvaru,Malleshappa N. Noolvi,Uttam A More,Sudipta Chakraborty,Ashutosh Dash,Tejraj M. Aminabhavi,Kumar P. Narayan,Vishnu Sutariya

Letter Article

Design and Synthesis of Novel 5-Arylisoxazole-1,3,4-thiadiazole Hybrids as α-Glucosidase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 5 Year: 2021 Page: 436-444
Author(s): Mina Saeedi,Azadeh Eslami,Seyedeh Sara Mirfazli,Mahsa Zardkanlou,Mohammad Ali Faramarzi,Mohammad Mahdavi,Tahmineh Akbarzadeh

Research Article

Design, Synthesis and Biological Evaluation of a Novel Series of Thiadiazole- Based Anticancer Agents as Potent Angiogenesis Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 15 Year: 2021 Page: 2041-2049
Author(s): Burcugül Altuğ-Tasa,Betül Kaya-Çavuşoğlu,Ayşe T. Koparal,Gülhan Turan,Ali S. Koparal,Zafer A. Kaplancıklı

Research Article

Evaluation of Biological Activity of Derivatives of 1,3,4-Thiadiazole, 1,3,4-Oxadiazole and 1,2,4-Triazole

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 21 Issue: 5 Year: 2021 Page: 905-911
Author(s): Gaurav M. Doshi,Mayuresh U. Bansode,Rakesh R. Somani

Mini-Review Article

2-Substituted-mercapto-quinazolin-4(3H)-ones as DHFR Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 21 Issue: 1 Year: 2021 Page: 2249-2260
Author(s): Hussein I. El-Subbagh,Mohamed A. Sabry

Review Article

Synthesis of N,N'-Diacylhydrazines and their Use in Various Synthetic Transformations

Journal: Current Organic Chemistry
Volume: 25 Issue: 1 Year: 2021 Page: 1394-1403
Author(s): Mohammed A. Baashen

Research Article

Antitubercular Potential of Novel Isoxazole Encompassed 1, 2, 4-Triazoles: Design, Synthesis, Molecular Docking Study and Evaluation of Antitubercular Activity

Journal: Anti-Infective Agents
Volume: 19 Issue: 2 Year: 2021 Page: 147-161
Author(s): Neenu Ganesh,Arun Kumar S,Manisha Singh,Venkaraddi Mangannavar Chandrashekar,Gurubasavaraj Veeranna Pujar

Mini-Review Article

Enoyl-Acyl Carrier Protein Reductase (INHA): A Remarkable Target to Exterminate Tuberculosis

Journal: Anti-Infective Agents
Volume: 19 Issue: 3 Year: 2021 Page: 252-266
Author(s): Surabhi Jain,Smriti Sharma,Dhrubo Jyoti Sen,Saurabh S Pandya

Research Article

Synthesis of Novel Aryl (4-Aryl-1h-Pyrrol-3-Yl) (Thiophen-2-Yl) Methanone Derivatives: Molecular Modelling, In Silico Admet, Anti-Inflammatory and Anti-Ulcer Activities

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 20 Issue: 2 Year: 2021 Page: 182-195
Author(s): Arif Pasha,Sumanta Mondal,Naresh Panigrahi

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