Search Result "S-mephenytoin"


An In Vitro, High Throughput, Seven CYP Cocktail Inhibition Assay for the Evaluation of New Chemical Entities Using LC-MS/MS

Journal: Drug Metabolism Letters
Volume: 5 Issue: 1 Year: 2011 Page: 17-24
Author(s): Jennifer N. Otten, Gary P. Hingorani, Dylan P. Hartley, Scott D. Kragerud, Ronald B. Franklin

High-Throughput, 384-Well, LC-MS/MS CYP Inhibition Assay Using Automation, Cassette-Analysis Technique and Streamlined Data Analysis

Journal: Drug Metabolism Letters
Volume: 5 Issue: 3 Year: 2011 Page: 220-230
Author(s): Jason S. Halladay, Erlie Marie Delarosa, Daniel Tran, Leslie Wang, Susan Wong, S. Cyrus Khojasteh

Research Article

A Novel In vitro Experimental System for the Evaluation of Enteric Drug Metabolism: Cofactor-Supplemented Permeabilized Cryopreserved Human Enterocytes (MetMax™ Cryopreserved Human Enterocytes)

Journal: Drug Metabolism Letters
Volume: 12 Issue: 2 Year: 2018 Page: 132-137
Author(s): Albert P. Li,Kirsten Amaral,Ming-Chih D. Ho

Evaluation of Cytochrome P450 Inhibition Assays Using Human Liver Microsomes by a Cassette Analysis /LC-MS/MS

Journal: Drug Metabolism Letters
Volume: 4 Issue: 3 Year: 2010 Page: 120-128
Author(s): Serenella Zambon, Stefano Fontana, Mahmud Kajbaf

Metabolism of R- and S-Warfarin by CYP2C19 into Four Hydroxywarfarins

Journal: Drug Metabolism Letters
Volume: 6 Issue: 3 Year: 2012 Page: 157-164
Author(s): So-Young Kim, Ji-Yeon Kang, Jessica H. Hartman, Sun-Ha Park, Drew R. Jones, Chul-Ho Yun, Gunnar Boysen, Grover P. Miller

Transcriptional Regulation of CYP2C19 and its Role in Altered Enzyme Activity

Journal: Current Drug Metabolism
Volume: 13 Issue: 8 Year: 2012 Page: 1196-1204
Author(s): Chakradhara Rao S. Uppugunduri, Youssef Daali, Jules Desmeules, Pierre Dayer, Maja Krajinovic, Marc Ansari

The Pharmacogenetics of CYP2C9 and CYP2C19: Ethnic Variation and Clinical Significance

Journal: Current Clinical Pharmacology
Volume: 2 Issue: 1 Year: 2007 Page: 93-109
Author(s): J. Rosemary, C. Adithan

Review Article

In vivo Phenotyping Methods: Cytochrome P450 Probes with Emphasis on the Cocktail Approach

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 1 Year: 2017 Page: 2035-2049
Author(s): Guillermo Alberto Keller,María Laura Ferreirós Gago,Roberto Alejandro Diez,Guillermo Di Girolamo

Assessment of Cytochrome P450 Induction in Human Hepatocytes Using the Cocktail Strategy Plus Liquid Chromatography Tandem Mass Spectrometry

Journal: Drug Metabolism Letters
Volume: 2 Issue: 3 Year: 2008 Page: 205-209
Author(s): Agustin Lahoz, Maria Teresa Donato, Laura Picazo, Jose V. Castell, Maria Jose Gomez-Lechon

Review Article

Use of Cocktail Probe Drugs for Indexing Cytochrome P450 Enzymes in Clinical Pharmacology Studies – Review of Case Studies

Journal: Drug Metabolism Letters
Volume: 13 Issue: 1 Year: 2019 Page: 3-18
Author(s): Poonam Giri,Harilal Patel,Nuggehally R. Srinivas

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