Search Result "Zolinza"


5-Aryl-1,3,4-Thiadiazole-Based Hydroxamic Acids as Histone Deacetylase Inhibitors and Antitumor Agents: Synthesis, Bioevaluation and Docking Study

Journal: Medicinal Chemistry
Volume: 11 Issue: 3 Year: 2015 Page: 296-304
Author(s): Tran Thi Lan Huong, Do Thi Mai Dung, Dao Thi Kim Oanh, Tran Thi Bich Lan, Phan Thi Phuong Dung, Vu Duc Loi, Kyung Rok Kim, Byung Woo Han, Jieun Yun, Jong Soon Kang, Youngsoo Kim, Sang-Bae Han, Nguyen-Hai Nam

New Benzothiazole/thiazole-Containing Hydroxamic Acids as Potent Histone Deacetylase Inhibitors and Antitumor Agents

Journal: Medicinal Chemistry
Volume: 9 Issue: 8 Year: 2013 Page: 1051-1057
Author(s): Truong Thanh Tung,Dao Thi Kim Oanh,Phan Thi Phuong Dung,Van Thi My Hue,Sang Ho Park,Byung Woo Han,Youngsoo Kim,Jin-Tae Hong,Sang-Bae Han,Nguyen-Hai Nam

Non-Cancer Uses of Histone Deacetylase Inhibitors: Effects on Infectious Diseases and β-Hemoglobinopathies+

Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 3 Year: 2009 Page: 272-291
Author(s): Dante Rotili, Giovanna Simonetti, Andrea Savarino, Anna T. Palamara, Anna R. Migliaccio, Antonello Mai

Epigenetic Regulation of Epithelial-Mesenchymal Transition by Hypoxia in Cancer: Targets and Therapy

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 10 Year: 2015 Page: 1272-1278
Author(s): Jian -Qiu Wang,Kou -Juey Wu

Editorial free to download

Epigenetic Modifications as Therapeutic Targets

Journal: Current Drug Targets
Volume: 21 Issue: 1 Year: 2020 Page: 1046-1046
Author(s): Si-Qi Feng,Yi-Chao Zheng

Commercially Available, FDA-approved Epigenetic Modifiers As Therapeutic Agents in Bacterial Infection

Journal: Clinical Anti-Inflammatory & Anti-Allergy Drugs (Discontinued)
Volume: 2 Issue: 1 Year: 2015 Page: 79-88
Author(s): Pádraic J. Dunne,Georgia Richard,Joseph Keane

Review Article

Designing Isoform-selective Inhibitors Against Classical HDACs for Effective Anticancer Therapy: Insight and Perspectives from In Silico

Journal: Current Drug Targets
Volume: 19 Issue: 7 Year: 2018 Page: 815-824
Author(s): Shabir Ahmad Ganai

Targeting Cancer with Epi-Drugs: A Precision Medicine Perspective

Journal: Current Pharmaceutical Biotechnology
Volume: 17 Issue: 10 Year: 2016 Page: 856-865
Author(s): Lisa Gherardini,Ankush Sharma,Enrico Capobianco,Caterina Cinti

Review Article

Recent Development of Novel HDAC6 Isoform-selective Inhibitors

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 2 Year: 2021 Page: 4133-4151
Author(s): Yunpeng Zhao,Tao Liang,Xuben Hou,Hao Fang

Review Article

Epigenetically Active Drugs Inhibiting DNA Methylation and Histone Deacetylation

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 8 Year: 2017 Page: 1167-1174
Author(s): Dimitry A. Chistiakov,Veronika A. Myasoedova,Alexander N. Orekhov,Yuri V. Bobryshev

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