Search Result "triazolo"


Research Article

Microwave-Assisted Regioselective Synthesis of Variously Functionalized [1,2,4]triazolo[3,4-b]quinazolin-5(1H)-ones

Journal: Current Organic Chemistry
Volume: 24 Issue: 1 Year: 2020 Page: 1892-1896
Author(s): Awad I. Said,Matti Haukka,Ferenc Fülöp

Research Article

A New Synthesis of Poly Heterocyclic Compounds Containing [1,2,4]triazolo and [1,2,3,4]tetrazolo Moieties and their DFT Study as Expected Anti-cancer Reagents

Journal: Current Organic Synthesis
Volume: 17 Issue: 3 Year: 2020 Page: 211-223
Author(s): El-sayed M. Abdelrehim,Doaa S. El-Sayed

Research Article

Design, Synthesis and Molluscicidal Activity of New Phosphorus Compounds Bearing Fluorine Substituted 1,2,4-Triazolo[3,2-c][1,2,4]triazine Derivatives

Journal: Letters in Organic Chemistry
Volume: 17 Issue: 3 Year: 2020 Page: 184-190
Author(s): Reda M. Abdel-Rahman,Abdulrahman S. Alharbi,Nawaa A. Alshammari,Yousuf O. Adnan

Research Article

DBU Catalysis: An Efficient Synthetic Strategy for 5,7-disubstituted-1,2,4- triazolo[1,5-a]pyrimidines

Journal: Current Organic Synthesis
Volume: 17 Issue: 1 Year: 2020 Page: 73-80
Author(s): Yogesh K. Pandey,Anu Mishra,Pratibha Rai,Jaya Singh,Jagdamba Singh,Ramendra K. Singh

Research Article

First Example of Antiparasitic Activity Influenced by Thermochromism: Leishmanicidal Evaluation of 5,7-dimethyl-1,2,4-triazolo[1,5-a]pyrimidine Metal Complexes

Journal: Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2020 Page: 422-430
Author(s): José M. Méndez-Arriaga,Itziar Oyarzabal,Álvaro Martín-Montes,Judith García-Rodríguez,Miguel Quirós,Manuel Sánchez-Moreno

Research Article

Directed Search of Anti-inflammatory Agents among (3HQuinazoline- 4-ylidene)hydrazides of N-protected Amino acids and their Heterocyclization Products

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2020 Page: 60-71
Author(s): Yulya Martynenko,Oleksii Antypenko,Inna Nosulenko,Galina Berest,Sergii Kovalenko

Research Article

In Vitro Biological Estimation of 1,2,3-Triazolo[4,5-d]pyrimidine Derivatives as Anti-breast Cancer Agent: DFT, QSAR and Docking Studies

Journal: Current Pharmaceutical Biotechnology
Volume: 21 Issue: 1 Year: 2020 Page: 70-78
Author(s): Oyebamiji A. Kolawole,Semire Banjo

Research Article

Design, Synthesis, Molecular Docking Study and Anti-Hepatocellular Carcinoma Evaluation of Some New Bis-Triazolothiadiazines

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 20 Issue: 9 Year: 2020 Page: 788-800
Author(s): Abdelaziz A. El-Sayed,Sobhi M. Gomha,Zeinab A. Muhammad,Elham Ezz El-Arab,Amira M. Elmetwally,Islam K. Matar

Research Article

Triazavirin - Potential Inhibitor for 2019-nCoV Coronavirus M Protease: A DFT Study

Journal: Current Molecular Medicine
Volume: 20 Issue: 0 Year: 2020 Page: 1-10
Author(s): Siyamak Shahab,Masoome Sheikhi

Research Article

A New Series of Triazolothiadiazines as Potential Anticancer Agents for Targeted Therapy of Non-small Cell Lung and Colorectal Cancers: Design, Synthesis, In Silico and In Vitro Studies Providing Mechanistic Insight into Their Anticancer Potencies

Journal: Medicinal Chemistry
Volume: 16 Issue: 0 Year: 2020 Page: 1-27
Author(s): Belgin Sever,Mehlika Dilek Altıntop,Gülşen Akalın Çiftçi,Ahmet Özdemir

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