Search Result "triazolo"


Review Article

Recent Advances of 1,2,4-triazolo[3,4-α]pyridines: Synthesis and Bioactivities

Journal: Current Organic Chemistry
Volume: 21 Issue: 16 Year: 2017 Page: 1626-1650
Author(s): Zhong-Hua Shen,Qiao Wang,Ming-Yan Yang,Zhao-Hui Sun,Jian-Quan Weng,Cheng-Xia Tan,Hong-Ke Wu,Liang Han,Xing-Hai Liu

Research Article

New Cyclopenta[4,5]pyrido[3,2:4,5]thieno[2,3-e][1,2,4]triazolo[4,3-c]pyrimidines and Cyclopenta[4,5]pyrido[3,2:4,5]thieno[2,3-e][1,2,4]triazolo[1,5-c]pyrimidines: Synthesis and Antimicrobial Activities

Journal: Current Organic Chemistry
Volume: 21 Issue: 1 Year: 2017 Page: 1227-1241
Author(s): Samvel N. Sirakanyan,Domenico Spinelli,Athina Geronikaki,Viktor A. Kartsev,Elmira K. Hakobyan,Henrik A. Panosyan,Hrachya M. Stepanyan,Luca Zuppiroli,Anush A. Hovakimyan

Research Article

Evaluation of the Novel Antichagasic Activity of [1,2,3]Triazolo[1,5-a]pyridine Derivatives

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 4 Year: 2017 Page: 399-411
Author(s): Michel Lapier,Maria C. Zuniga-Lopez,Benjamin Aguilera-Venegas,Rosa Adam,Belen Abarca,Rafael Ballesteros,Rodrigo Lopez-Munoz,Juan Diego Maya,Claudio Olea-Azar

Review Article

Leishmanicidal and Trypanocidal Activity of Metal Complexes with 1,2,4-Triazolo[1,5-a]pyrimidines: Insights on their Therapeutic Potential against Leishmaniasis and Chagas Disease

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 25 Year: 2017 Page: 2796-2806
Author(s): Juan M. Salas,Ana B. Caballero,Ginés M. Esteban-Parra,José M. Méndez-Arriaga

Letter Article

Genotoxicity of 4-(piperazin-1-yl)-8-(trifluoromethyl)pyrido[2,3-e][1,2,4] triazolo[4,3-a]pyrazine, a Potent H4 Receptor Antagonist for the Treatment of Allergy: Evidence of Glyoxal Intermediate Involvement

Journal: Drug Metabolism Letters
Volume: 11 Issue: 2 Year: 2017 Page: 144-148
Author(s): Mithat Gunduz,Amanda L. Cirello,Peter Klimko,Jennifer L. Dumouchel,Upendra A. Argikar

Research Article

Novel [1,2,4] Triazol [4,3-a] Pyridine Derivatives as Potential Selective c-Met Inhibitors with Improved Pharmacokinetic Properties

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 8 Year: 2017 Page: 1102-1112
Author(s): Junjun Zhao,Shaohua Gou,Xiaobing Zhang,Yan Liang,Lei Fang

Review Article

Searching for Novel Janus Kinase-2 Inhibitors Using a Combination of Pharmacophore Modeling, 3D-QSAR Studies and Virtual Screening

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 268-294
Author(s): Eleni Vrontaki,Georgia Melagraki,Antreas Afantitis,Thomas Mavromoustakos,George Kollias

Review Article

1,N6-ethenoadenine and other Fluorescent Nucleobase Analogs as Substrates for Purine-Nucleoside Phosphorylases: Spectroscopic and Kinetic Studies

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 4 Year: 2017 Page: 6948-6966
Author(s): Jacek Wierzchowski,Alicja Stachelska-Wierzchowska,Beata Wielgus-Kutrowska,Agnieszka Bzowska

Research Article

Synthesis, EGFR Inhibition and Anti-cancer Activity of New 3,6-dimethyl-1-phenyl-4-(substituted-methoxy)pyrazolo[3,4-d] pyrimidine Derivatives

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 10 Year: 2017 Page: 1389-1400
Author(s): Rania B. Bakr,Ahmed B. M. Mehany,Khaled R. A. Abdellatif

Review Article

Dimroth Rearrangement-Old but not Outdated

Journal: Current Organic Chemistry
Volume: 21 Issue: 25 Year: 2017 Page: 2515-2529
Author(s): Anna Krajczyk,Jerzy Boryski

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