Search Result "topoisomerase I"


Synthesis and Biological Evaluation of Pyrazolo[3,4-b]pyridin-4-ones as a New Class of Topoisomerase II Inhibitors

Journal: Medicinal Chemistry
Volume: 11 Issue: 4 Year: 2015 Page: 342-353
Author(s): Mojgan Aghazadeh Tabrizi,Pier Giovanni Baraldi,Stefania Baraldi,Filippo Prencipe,Delia Preti,Giulia Saponaro,Romeo Romagnoli,Stefania Gessi,Stefania Merighi,Angela Stefanelli,Debora Fazzi,Pier Andrea Borea,Rodolfo Couto Maia,Nelilma C. Romeiro,Carlos A. M. Fraga,Eliezer J. Barreiro

Mannich Base Derivatives as the Potential Candidates of Human Topoisomerase II Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 12 Issue: 2 Year: 2015 Page: 103-108
Author(s): Huseyin Istanbullu, Muge Senarisoy, Ercin Erciyas, Zeki Topcu

11-Phenylundeca-5Z,9Z-dienoic Acid: Stereoselective Synthesis and Dual Topoisomerase I/IIα Inhibition

Journal: Current Cancer Drug Targets
Volume: 15 Issue: 6 Year: 2015 Page: 504-510
Author(s): Vladimir A. D’yakonov,Lilya U. Dzhemileva,Aleksey A. Makarov,Alfiya R. Mulyukova,Dmitry S. Baevd,Elza K. Khusnutdinova,Tatiana G. Tolstikova,Usein M. Dzhemilev

Anti-Tubercular Agents from Glycyrrhiza glabra

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 11 Year: 2015 Page: 1043-1049
Author(s): Komal Kalani,Vinita Chaturvedi,Sarfaraz Alam,Feroz Khan,Santosh Kumar Srivastava

Crystallographic Study and Biological Evaluation of 1,4-dimethyl-N-alkylcarbazoles†

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 11 Year: 2015 Page: 973-979
Author(s): Carmela Saturnino,Anna Caruso,Pasquale Longo,Anna Capasso,Attilio Pingitore,Maria Cristina Caroleo,Erika Cione,Mariarita Perri,Francesco Nicolo,Viviana Mollica Nardo,Luigi Monsu Scolaro,Maria Stefania Sinicropi,Maria Rosaria Plutino,Hussein El-Kashef

Recent Developments on Thiourea Based Anticancer Chemotherapeutics

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 15 Issue: 2 Year: 2015 Page: 163-175
Author(s): Vikas Kumar,Swapandeep Singh Chimni

Potential Therapeutic Advantages of Doxorubicin when Activated by Formaldehyde to Function as a DNA Adduct-Forming Agent

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 14 Year: 2015 Page: 1409-1422
Author(s): Suzanne M. Cutts,Ada Rephaeli,Abraham Nudelman,Michal Ugarenko,Don R. Phillips

Design, Synthesis and Evaluation of Novel 9-substituted Carbazole Derivatives as Potential Anticancer Agents

Journal: Letters in Drug Design & Discovery
Volume: 12 Issue: 9 Year: 2015 Page: 760-765
Author(s): Nitin Kumar,Devender Pathak

Combination Therapy of Intraperitoneal Rapamycin and Convection- Enhanced Delivery of Nanoliposomal CPT-11 in Rodent Orthotopic Brain Tumor Xenografts

Journal: Current Cancer Drug Targets
Volume: 15 Issue: 4 Year: 2015 Page: 352-362
Author(s): Marina Mendiburu-Elicabe,Jon Gil-Ranedo

Neocryptolepine: A Promising Indoloisoquinoline Alkaloid with Interesting Biological Activity. Evaluation of the Drug and its Most Relevant Analogs

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 17 Year: 2015 Page: 1683-1707
Author(s): Enrique L. Larghi,Andrea B. J. Bracca,Abel A. Arroyo Aguilar,Daniel A. Heredia,Jorgelina L. Pergomet,Sebastian O. Simonetti,Teodoro S. Kaufman

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