Search Result "tofacitinib"


Review Article

Tofacitinib, an Oral Janus Kinase Inhibitor: Perspectives in Dermatology

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 1 Year: 2017 Page: 1158-1167
Author(s): Kresimir Kostovic,Sandra J. Gulin,Zrinka B. Mokos,Romana Ceovic

Review Article open access plus

A Systematic Analysis of Physicochemical and ADME Properties of All Small Molecule Kinase Inhibitors Approved by US FDA from January 2001 to October 2015

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 29 Year: 2017 Page: 3159-3184
Author(s): Zhihong O`Brien,Mehran F. Moghaddam

Review Article

Pyrrolo[2,3-d]Pyrimidines as Kinase Inhibitors

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 19 Year: 2017 Page: 2059-2085
Author(s): Francesca Musumeci,Monica Sanna,Giancarlo Grossi,Chiara Brullo,Anna Lucia Fallacara,Silvia Schenone

Review Article

Old But Good: Modified-Release Prednisone in Rheumatoid Arthritis

Journal: Reviews on Recent Clinical Trials
Volume: 12 Issue: 2 Year: 2017 Page: 124-128
Author(s): Francesco Ursini, Saverio Naty, Caterina Bruno, Rosa Daniela Grembiale

Review Article

Protein Kinases as Drug Targets in Human and Animal Diseases

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 2 Year: 2017 Page: 99-106
Author(s): Suvarna G. Kini, Vikas Garg, Sharada Prasanna, Revathi Rajappan, Muhammad Mubeen

Review Article

Safety of Systemic Biologic Agents in the Treatment of Non-malignant Skin Disorders

Journal: Current Drug Safety
Volume: 12 Issue: 2 Year: 2017 Page: 76-94
Author(s): George Badavanis,Efstathia Pasmatzi,Alexandra Monastirli,Dionysios Tsambaos

Review Article

Specificity of Binding in Protein Kinases

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 2 Year: 2017 Page: 89-98
Author(s): Satya P. Gupta, Basheerulla Shaik, Vijay K. Agrawal

Review Article

Searching for Novel Janus Kinase-2 Inhibitors Using a Combination of Pharmacophore Modeling, 3D-QSAR Studies and Virtual Screening

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 268-294
Author(s): Eleni Vrontaki,Georgia Melagraki,Antreas Afantitis,Thomas Mavromoustakos,George Kollias

Proteomics in the Characterization of New Target Therapies in Pediatric Obesity Treatment

Ebook: Anti-Obesity Drug Discovery and Development

Volume: 3 Year: 2017
Author(s): Gillian E. Walker,Marilisa De Feudis,Marta Roccio,Gianni Bona,Flavia Prodam
Doi: 10.2174/9781681081878117030005
Review Article

Leveraging Structural Diversity and Allosteric Regulatory Mechanisms of Protein Kinases in the Discovery of Small Molecule Inhibitors

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 4 Year: 2017 Page: 4838-4872
Author(s): Gennady M. Verkhivker

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