Search Result "thiazolidinones"


Research Article

Synthesis and Biological Evaluation of New 4-Thiazolidinone Derivatives as Carbonic Anhydrase Inhibitors

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 2 Year: 2017 Page: 80-85
Author(s): Hayriye Genc,Busra Ceken,Cigdem Bilen,Zubeyde Sackes,Nahit Gencer,Oktay Arslan

Research Article

Synthesis, ADME Evaluation, and In Vitro Antimycobacterial Studies of a Novel Series of 2-Thiazolylimino-5-Arylidene-4-Thiazolidinone Derivatives

Journal: Anti-Infective Agents
Volume: 15 Issue: 1 Year: 2017 Page: 38-44
Author(s): Alka Mital,Rohani Prasad Burman,Rajesh Gour,Sarbjit Singh Jhamb,Manjinder Singh Gill

Research Article

Molecular Docking, Molecular Dynamics, and In Silico Prediction of the Toxic Potential of Primaquine Thiazolidinone Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 3 Year: 2017 Page: 345-353
Author(s): Erika Murce,Andre Silva Pimentel

Research Article

Thiazolidinone Constraint Combretastatin Analogs as Novel Antitubulin Agents: Design, Synthesis, Biological Evaluation and Docking Studies

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 2 Year: 2017 Page: 230-240
Author(s): Sahil Sharma,Manish Kumar Gupta,Ajit Kumar Saxena,Preet Mohinder Singh Bedi

Research Article

Synthesis and Antimicrobial Activity Evaluation of the Pyrrole-Derived Heterocycles Bearing Two Functionalities

Journal: Current Organic Synthesis
Volume: 14 Issue: 1 Year: 2017 Page: 137-142
Author(s): Wael S.I. Abou-Elmagd,Ahmed Abdel Aziz,Ahmed I. Hashem

Research Article

Microwave Assisted and Efficient Synthesis of Substituted Thiazole Acid Derivatives

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 7 Year: 2017 Page: 517-524
Author(s): Dattatraya N. Pansare,Rohini N. Shelke,Chandrakant D. Pawar

Research Article

Antimicrobial and Cytotoxicity Activities of 2-(aryl)-3-(benzo[d][1,3] dioxol-5-yl)thiazolidin-4-ones

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 9 Year: 2017 Page: 1042-1047
Author(s): Silvana P. Souza,Hellen G. Masteloto,Daniel S. da Silva,Juliana H. Azambuja,Elizandra Braganhol,Juliana S. Ribeiro,Rafael G. Lund,Wilson Cunico

Review Article

HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: SAR and Lead Optimization Using CoMFA and CoMSIA Studies (1995-2016)

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 34 Year: 2017 Page: 3774-3812
Author(s): Murugesan Vanangamudi,Vasanthanathan Poongavanam,Vigneshwaran Namasivayam

Research Article

Structure-Based Hybridization, Conventional and Microwave Irradiated Synthesis, Biological Evaluation and Molecular Docking Studies of New Compounds Derived from Thiomorpholin

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 4 Year: 2017 Page: 444-463
Author(s): Serpil Demirci,Fatma Aksakal,Nesrin Colak,Serdar Ulker,Ahmet Demirbas,Neslihan Demirbas

Research Article

Quorum Sensing Inhibitor Activities of Celecoxib Derivatives in Pseudomonas aeruginosa

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 5 Year: 2017 Page: 613-618
Author(s): Seyhan Ulusoy,Sevil Senkardes,Inci Coskun,Gulgun Bosgelmez-Tınaz,Laurent Soulere,Yves Queneau,S. Guniz Kucukguzel

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