Search Result "thiadiazoles"


Novel 1,2,4-Triazolo[3,4-b]-1,3,4-thiadiazole Derivatives as Dual Analgesic/Anti-inflammatory and Antimicrobial Agents

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 2 Year: 2012 Page: 204-212
Author(s): Birsen Tozkoparan, Sevim Peri Aytac, Sule Gursoy, Selami Gunal, Goknur Aktay

Synthesis, Docking and Biological Evaluation of Some Novel 5-bromo-2- (5-aryl-1,3,4-thiadiazol-2-yl)isoindoline-1,3-dione Derivatives Targeting ATP-binding Site of Topoisomerase II

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 7 Year: 2012 Page: 668-675
Author(s): Ankur Gupta,Priya Singh,Bhagyashree Kamble,Aditi Kulkarni,Moola Joghee Nanjan Chandrasekar

Synthesis of Novel Quinolone and Coumarin Based 1,3,4-Thiadiazolyl and 1,3,4-Oxadiazolyl N-Mannich Bases as Potential Antimicrobials

Journal: Letters in Organic Chemistry
Volume: 9 Issue: 7 Year: 2012 Page: 478-486
Author(s): Rahul V. Patel,Jigar K. Patel,Premlata Kumari,Kishor H. Chikhalia

Synthesis of Novel Azetidinone Derivatives as Antitubercular Agents

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 6 Year: 2012 Page: 611-617
Author(s): M. Himaja,Asif Karigar,M. V. Ramana,D. Munirajasekhar,Mukesh S. Sikarwar

Microwave Assisted Synthesis of Five Membered Azaheterocyclic Systems

Journal: Current Organic Chemistry
Volume: 16 Issue: 6 Year: 2012 Page: 789-828
Author(s): Rajeev Sakhuja, Siva S. Panda, Kiran Bajaj

Novel Biotransformation Process of Podophyllotoxin to 4 -Sulfur-Substituted Podophyllum Derivates with Anti-Tumor Activity by Penicillium purpurogenum Y.J. Tang

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 6 Year: 2012 Page: 927-936
Author(s): J.-K. Bai, W. Zhao, H.-M. Li, Y.-J. Tang

A Study on the Biological Activity of 2-thioxo-imidazolidin-4-ones

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 5 Year: 2012 Page: 549-555
Author(s): Sudha Vengurlekar, Rajesh Sharma, Piyush Trivedi

Graphical Abstracts

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 7 Year: 2012 Page: i-iv
Author(s):

Graphical Abstracts

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 2 Year: 2012 Page: i-iv
Author(s):

The Bioisosteric Concept Applied to Cannabinoid Ligands

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 28 Year: 2012 Page: 4794-4815
Author(s): C. Mugnaini,S. Pasquini,F. Corelli

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