Search Result "tacrine"


Synthesis and Biological Activity of New 2,3-dihydro-1H-cyclopenta[b]- quinoline Derivatives as Acetylcholinesterase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 7 Year: 2012 Page: 645-654
Author(s): Pawel Szymanski,Magdalena Markowicz,Marek Bajda,Barbara Malawska,Elzbieta Mikiciuk-Olasik

Acetylcholinesterase Inhibitors as Pretreatment Before Acute Exposure to Organophosphates: Assessment Using Methyl-Paraoxon

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 11 Issue: 8 Year: 2012 Page: 1052-1060
Author(s): Dietrich E. Lorke,Mohamed Y. Hasan,Syed M. Nurulain,Mohamed Shafiullah,Kamil Kuca,Georg A. Petroianu

QSAR Applications During Last Decade on Inhibitors of Acetylcholinesterase in Alzheimer’s Disease

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 10 Year: 2012 Page: 936-946
Author(s): K. Y. Wong,P. R. Duchowicz,A. G. Mercader,E. A. Castro

Designed Multiple Ligands: Basic Research vs Clinical Outcomes

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 20 Year: 2012 Page: 3353-3387
Author(s): L. Costantino,D. Barlocco

Design, Synthesis and Biological Evaluation of Scutellarein Derivatives as Potential Anti-Alzheimers Disease Candidates Based on Metabolic Mechanism

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 1 Year: 2012 Page: 78-83
Author(s): Shu-Lin Song, Nian-Guang Li, Yu-Ping Tang, Zhen-Jiang Wang, Li-Hua Qian, Hao Tang, Jin-Ao Duan

The Metabolic Rationale for a Lack of Cross-reactivity Between Sulfonamide Antimicrobials and Other Sulfonamide-containing Drugs

Journal: Drug Metabolism Letters
Volume: 6 Issue: 2 Year: 2012 Page: 129-133
Author(s): David F. Lehmann

Iontophoresis: Drug Delivery System by Applying an Electrical Potential Across the Skin

Journal: Drug Delivery Letters
Volume: 2 Issue: 4 Year: 2012 Page: 270-280
Author(s): Tarun Garg, Amit Kumar Goyal

Ladostigil: A Novel Multimodal Neuroprotective Drug with Cholinesterase and Brain-Selective Monoamine Oxidase Inhibitory Activities for Alzheimers Disease Treatment

Journal: Current Drug Targets
Volume: 13 Issue: 4 Year: 2012 Page: 483-494
Author(s): Orly Weinreb, Tamar Amit, Orit Bar-Am, Moussa B.H. Youdim

An Overview on Potential Neuroprotective Compounds for Management of Alzheimer’s Disease

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 11 Issue: 8 Year: 2012 Page: 1006-1011
Author(s): Ishfaq Ahmed Sheikh,Riyasat Ali,Tanveer A. Dar,Mohammad Amjad Kamal

CNS Drug Development – Lost in Translation?

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 10 Year: 2012 Page: 959-970
Author(s): A. Talevi,C. L. Bellera,M. Di Ianni,M. Gantner,L. E. Bruno-Blanch,. A. Castro

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