Search Result "submicromolar"


Antileishmanial and Antimalarial Chalcones: Synthesis, Efficacy and Cytotoxicity of Pyridinyl and Naphthalenyl Analogs

Journal: Medicinal Chemistry
Volume: 3 Issue: 2 Year: 2007 Page: 115-119
Author(s): C. E. Gutteridge, J. V. Vo, C. B. Tillett, J. A. Vigilante, J. R. Dettmer, S. L. Patterson, K. A. Werbovetz, J. Capers, D. A. Nichols, A. K. Bhattacharjee, L. Gerena

Azetidine-Based Inhibitors of Dipeptidyl Peptidase IV (DPP IV)

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 6 Year: 2007 Page: 597-608
Author(s): Dana Ferraris, Sergei Belyakov, Weixing Li, Eddie Oliver, Yao-Sen Ko, David Calvin, Susan Lautar, Bert Thomas, Camilo Rojas

Metabolism of Sanguinarine: The Facts and The Myths

Journal: Current Drug Metabolism
Volume: 8 Issue: 2 Year: 2007 Page: 173-176
Author(s): Z. Dvorak, V. Simanek

Recent Developments in Cholinesterases Inhibitors for Alzheimers Disease Treatment

Journal: Current Medicinal Chemistry
Volume: 14 Issue: 2 Year: 2007 Page: 2654-2679
Author(s): Anna Musial, Marek Bajda, Barbara Malawska

BACE Inhibitors as Potential Therapeutics for Alzheimers disease

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 2 Issue: 3 Year: 2007 Page: 188-199
Author(s): Genevieve Evin, Vijaya B. Kenche

Protein-Protein Interaction Inhibitors: Small Molecules from Screening Techniques

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2007 Page: 922-927
Author(s): Steven Fletcher, Andrew D. Hamilton

Small Molecule Inhibitors of the XIAP Protein-Protein Interaction

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2007 Page: 966-971
Author(s): Hemaka A. Rajapakse

Validated Ligand Binding Sites in CCK Receptors. Next Step: Computer-Aided Design of Novel CCK Ligands

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2007 Page: 1243-1247
Author(s): Irina G. Tikhonova, Esther Marco, Elodie Lahlou-Archer, Ingrid Langer, Magali Foucaud, Bernard Maigret, Daniel Fourmy

Novel, Acidic CCR2 Receptor Antagonists: From Hit to Lead

Journal: Letters in Drug Design & Discovery
Volume: 4 Issue: 3 Year: 2007 Page: 185-191
Author(s): D. Zou, H.-X. Zhai, J. Eckman, P. Higgins, M. Gillard, L. Knerr, S. Carre, P. Pasau, P. Collart, J. Grassi

Oncogenic Fusion Tyrosine Kinases as Molecular Targets for Anti-Cancer Therapy

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 7 Issue: 6 Year: 2007 Page: 594-611
Author(s): Rosalind H. Gunby, Elisa Sala, Carmen J. Tartari, Miriam Puttini, Carlo Gambacorti-Passerini, Luca Mologni

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