Search Result "submicromolar"


Research Article

PARG Inhibitors and Functional PARG Inhibition Models

Journal: Current Protein & Peptide Science
Volume: 17 Issue: 7 Year: 2016 Page: 641-653
Author(s): Yuka Sasaki, Miyuki Hozumi, Hiroaki Fujimori, Yasufumi Murakami, Fumiaki Koizumi, Kengo Inoue, Mitsuko Masutani

The NOX1/4 Inhibitor GKT136901 as Selective and Direct Scavenger of Peroxynitrite

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 3 Year: 2014 Page: 365-376
Author(s): S. Schildknecht,A. Weber,H. R. Gerding,R. Pape,M. Robotta,M. Drescher,A. Marquardt,A. Daiber,B. Ferger,M. Leist

Disaggregation of Tau as a Therapeutic Approach to Tauopathies

Journal: Current Alzheimer Research
Volume: 7 Issue: 3 Year: 2010 Page: 235-240
Author(s): K. Duff, J. Kuret, E.E Congdon

New Potent and Selective Inhibitor of Pim-1/3 Protein Kinases Sensitizes Human Colon Carcinoma Cells to Doxorubicin

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 14 Issue: 9 Year: 2014 Page: 1228-1236
Author(s): Pascale Moreau,Lyubov G. Dezhenkova,Fabrice Anizon,Lionel Nauton,Vincent Thery,Shuguang Liang,Dmitry N. Kaluzhny,Alexander A. Shtil

Research Article

The Oxime Derivatives of 1-R-1H-Naphtho[2,3-d][1,2,3]triazole-4,9-dione 2-oxides: Synthesis and Properties

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 1814-1823
Author(s): Leonid M. Gornostaev,Vladimir B. Tsvetkov,Alina A. Markova,Tatyana I. Lavrikova,Yulia G. Khalyavina,Anastasia S. Kuznetsova,Dmitry N. Kaluzhny,Alexei V. Shunayev,Maria V. Tsvetkova,Valeria A. Glazunova,Vladimir V. Chernyshev,Alexander A. Shtil

Review Article

The Syntheses and Medicinal Attributes of Phenanthrenes as AnticancerAgents: A Quinquennial Update

Journal: Current Medicinal Chemistry
Volume: 29 Issue: 2 Year: 2022 Page: 3530-3556
Author(s): Nagula Shankaraiah,Sayali Mone,Kritika Laxmikeshav,Sarthak Jhingran

Research Article

Sulphur-Containing Heterocycles as Antimycobacterial Agents: Recent Advances in Thiophene and Thiadiazole Derivatives

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 2921-2952
Author(s):

Research Article

Synthesis, Cytotoxicity, Anti-migration and Anti-invasion Activity of Diphyllin Heterocyclic Derivatives

Journal: Medicinal Chemistry
Volume: 17 Issue: 0 Year: 2021 Page: 1-9
Author(s): Weidong Shen,Haijiao Chen,Miaomiao Wu,Ting Zhang,Li Zhu,Yu Zhao

Applications of Adenosine Receptor Ligands in Medical Imaging by Positron Emission Tomography

Journal: Current Pharmaceutical Design
Volume: 8 Issue: 2 Year: 2002 Page: 2345-2352
Author(s): Marcus H. Holschbach, Ray A. Olsson

Research Article

Selective Cytotoxic Effects of 5-Trifluoromethoxy-1H-indole-2,3-dione 3-ThiosemicarbazoneDerivatives on Lymphoid-originated Cells

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 22 Issue: 2 Year: 2022 Page: 349-355
Author(s): Ferdane Danışman-Kalındemirtaş,Serap Erdem-Kuruca,Kadriye Akgün-Dar,Zeynep Karakaş,Özge Soylu,Nilgün Karali

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