Search Result "structure-inhibition relationship"


Review Article

Quantitative Structure-Activity Relationship Studies: Understanding the Mechanism of Tyrosine Kinase Inhibition

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 2 Year: 2017 Page: 139-159
Author(s): Vaishali M. Patil, Satya P Gupta, Neeraj Masand

Research Article

Synthesis and Structure-activity Relationships of Chalcone Derivatives as Inhibitors of Ovarian Cancer Cell Growth

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 11 Year: 2017 Page: 1259-1266
Author(s): Zachary D. Tucker,Francis J. Barrios,Amanda J. Krzysiak

Review Article

Understanding the Structural Basis for Inhibition of Cyclin-Dependent Kinases. New Pieces in the Molecular Puzzle

Journal: Current Drug Targets
Volume: 18 Issue: 9 Year: 2017 Page: 1104-1111
Author(s): Nayara M. Bernhardt Levin, Val Oliveira Pintro, Mauricio Boff de Avila, Bruna Boldrini de Mattos, Walter Filgueira De Azevedo Jr.

Research Article

In vitro α-Glucosidase Inhibition by Non-sugar based Triazoles of Dibenzoazepine, their Structure-Activity Relationship, and Molecular Docking

Journal: Medicinal Chemistry
Volume: 13 Issue: 7 Year: 2017 Page: 698-704
Author(s): Maria A. Khan,Kulsoom Javaid,Abdul Wadood,Alam Jamal,Farhana Batool,Saba Fazal-ur-Rehman,Fatima Z. Basha,Muhammad I. Choudhary

Research Article

Quantitative Structure-Activity Relationship and Docking Studies on a Series of Oxadiazole and Triazole Substituted Naphthyridines as HIV-1 Integrase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 10-27
Author(s): Basheerulla Shaik,Vijay Agrawal,Satya P. Gupta,Urvana Menon

Review Article

Pregnancy-Specific β1-Glycoproteins: Combined Biomarker Roles, Structure/Function Relationships and Implications for Drug Design

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 3 Year: 2017 Page: 245-267
Author(s): Nurbubu T. Moldogazieva,Innokenty M. Mokhosoev,Alexander A. Terentiev

Review Article

Structure-activity Relationship Studies of New Marine Anticancer Agents and their Synthetic Analogues

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 4 Year: 2017 Page: 4779-4799
Author(s): Sergey N. Fedorov,Valentin A. Stonik,Friedemann Honecker,Sergey A. Dyshlovoy

Review Article

Isoquinoline Alkaloids and Their Antiviral, Antibacterial, and Antifungal Activities and Structure-activity Relationship

Journal: Current Organic Chemistry
Volume: 21 Issue: 18 Year: 2017 Page: 1920-1934
Author(s): Zhi-Xing Qing,Peng Yang,Qi Tang,Pi Cheng,Xiu-Bin Liu,Ya-jie Zheng,Yi-Song Liu,Jian-Guo Zeng

Cardioprotective Plant Alkaloids: Ethnopharmacology, Structure Activity Relationship and Synthetic Analogues

Ebook: Herbal Medicine Back to the Future

Volume: 1 Year: 2017
Author(s): Abhijit Dey,Samapika Nandy,Anuradha Mukherjee,Rabindranath Bhattacharyya
Doi: 10.2174/9781681084893117010009
Research Article

Molecular Docking and Structure Activity Relationship Studies of NSAIDs. What do they Reveal about IC50?

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 8 Year: 2017 Page: 949-958
Author(s): Chrysoula Mikra,Georgios Rossos,Sotirios K. Hadjikakou,Nikolaos Kourkoumelis

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