Search Result "serine/threonine protein kinases"


Conformationally Constrained Peptides as Protein Tyrosine Kinase Inhibitors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2852-2866
Author(s): Rakesh K. Tiwari,Keykavous Parang

Synthesis of Cis-Fused Pyran Indolocarbazole Derivatives that Inhibit FLT3 Kinase and the DNA Damage Kinase, Checkpoint Kinase 1

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 12 Issue: 3 Year: 2012 Page: 194-201
Author(s): Francoise M. Perron-Sierra, Nathalie Kucharkzyk, Celine Boucley, Christel Guyard-Daumas, Sophie Sciberras, Christine Fouache, Sabine Plantier, Aurelie Studeny, Celine Bossard, Patrick J. Casara, Roy M. Golsteyn

Exploiting Substrate Recognition for Selective Inhibition of Protein Kinases

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2914-2920
Author(s): Avital Licht-Murava,Hagit Eldar-Finkelman

Targeting Protein Kinases in the Malaria Parasite: Update of an Antimalarial Drug Target

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2012 Page: 456-472
Author(s): Veronica M. Zhang, Marina Chavchich, Norman C. Waters

Structural and Functional Relationships Between GSK3α and GSK3β Proteins

Journal: Current Biotechnology
Volume: 1 Issue: 1 Year: 2012 Page: 80-87
Author(s): C. Laura Sayas, Jeronimo Jurado, Jesus Avila, Nieves Villanueva

Polo-Like Kinases Inhibitors

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2012 Page: 3937-3948
Author(s): L. Garuti, M. Roberti, G. Bottegoni

New Directions in Targeting Protein Kinases: Focusing Upon True Allosteric and Bivalent Inhibitors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2936-2945
Author(s): Vandana Lamba,Indraneel Ghosh

Yeast as a Powerful Model System for the Study of Apoptosis Regulation by Protein Kinase C Isoforms

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 17 Year: 2012 Page: 2492-2500
Author(s): Rui D. Silva,Lucilia Saraiva,Isabel Coutinho,Jorge Goncalves,Manuela Corte-Real

Protein Kinase C-theta Inhibitors: A Novel Therapy for Inflammatory Disorders

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 30 Year: 2012 Page: 4725-4746
Author(s): Sukhvir Chand,Nisha Mehta,Malkeet Singh Bahia,Anshuman Dixit,Om Silakari

Small Molecule Kinase Inhibitors as Anti-Cancer Therapeutics

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2012 Page: 399-411
Author(s): O. Chahrour,D. Cairns,Z. Omran

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