Search Result "receptor biased agonism"


Small Molecule Antagonists of Integrin Receptors

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 2 Year: 2010 Page: 2371-2392
Author(s): A. Perdih, M. Sollner Dolenc

Understanding Functional Residues of the Cannabinoid CB1 Receptor for Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 8 Year: 2010 Page: 779-798
Author(s): Joong-Youn Shim

Emerging Opportunities and Concerns for Drug Discovery at Serotonin 5-5-HT2B Receptors

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 5 Year: 2010 Page: 493-503
Author(s): Jose Brea, Julio Castro-Palomino, Sandra Yeste, Elena Cubero, Antonio Parraga, Eduardo Dominguez, Maria Isabel Loza

Targeting Platelet G-Protein Coupled Receptors (GPCRs): Looking Beyond Conventional GPCR Antagonism

Journal: Current Vascular Pharmacology
Volume: 8 Issue: 2 Year: 2010 Page: 140-154
Author(s): Louisa Dowal, Robert Flaumenhaft

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 8 Year: 2010 Page: 768-778
Author(s): Charles A. Lunn

Pathway-Specific, Species, and Sub-Type Counterscreening for Better GPCR Hits in High Throughput Screening

Journal: Current Pharmaceutical Biotechnology
Volume: 11 Issue: 7 Year: 2010 Page: 757-763
Author(s): Robert Swanson, James R. Beasley

High Content Screening of CXCR2-Dependent Signalling Pathways

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 13 Issue: 1 Year: 2010 Page: 3-15
Author(s): Michael Wolff, Simone Krede, Dorothea Haasen, Jorg Wiedenmann, G. Ulrich Nienhaus, Barbara Kistler, Franz Oswald, Ralf Heilker

Clinical Trials for Neuroprotection in ALS

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 9 Issue: 3 Year: 2010 Page: 305-313
Author(s): G. Siciliano, C. Carlesi, L. Pasquali, S. Piazza, S. Pietracupa, F. Fornai, S. Ruggieri, L. Murri

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