Search Result "pyrimidine derivatives"


Review Article

The Chemistry and Bio-Medicinal Significance of Pyrimidines & Condensed Pyrimidines

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 3133-3174
Author(s): K. S. Jain, N. Arya, N. N. Inamdar, P. B. Auti, S. A. Unawane, H. H. Puranik, M. S. Sanap, A. D. Inamke, V. J. Mahale, C. S. Prajapati, C. J. Shishoo

Review Article

Pyrimidine-fused Derivatives: Synthetic Strategies and Medicinal Attributes

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 3175-3210
Author(s): Gaurav Joshi, Himanshu Nayyar, Jimi Marin Alex, Gajendra S. Vishwakarma, Sunil Mittal, Raj Kumar

Research Article

Microwave Assisted Synthesis, Biological Characterization and Docking Studies of Pyrimidine Derivatives

Journal: Current Microwave Chemistry
Volume: 3 Issue: 3 Year: 2016 Page: 178-186
Author(s): Sanjay K. Rathwa,Manoj N. Bhoi,Mayuri A. Borad,Kinjal D. Patel,Dhanji P. Rajani,Smita D. Rajani,Hitesh D. Patel

Enzymology of Pyrimidine Metabolism and Neurodegeneration

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 14 Year: 2016 Page: 1408-1431
Author(s): Silvia Vincenzetti,Valeria Polzonetti,Daniela Micozzi,Stefania Pucciarelli

Research Article

Synthesis of Some Novel 5,7-Disubstituted-2-phenyl-5H-[1,3,4]thiadiazolo [3,2-a]pyrimidine Derivatives and Evaluation of Their Biological Activity

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 9 Year: 2016 Page: 661-671
Author(s): Talavara Venkatesh,Yadav D. Bodke,Nibin M. Joy,B. M. Vinoda,Yallappa Shiralgi,B. L. Dhananjaya

Research Article

Topomer CoMFA 3D-QSAR and Docking Studies of Pyrimidine Inhibitors of Pneumocystis Carinii Dihydrofolate Reductase

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 1 Year: 2016 Page: 1055-1062
Author(s): Jianbo Tong, Pei Zhan, Tuanli Yao, Lanbing Ma, Min Bai

Research Article

Synthesis and In Vitro Activity of Pyrrolo[3,4-d]pyrimidine-2,5-diones as Potential Non-nucleoside HCV Inhibitors

Journal: Current Enzyme Inhibition
Volume: 12 Issue: 2 Year: 2016 Page: 170-176
Author(s): Amany S. Mostafa, Serry A. El Bialy, Waleed A. Bayoumi, Youki Ueda, Masanori Ikeda, Nobuyuki Kato, Ali M. Abdelal

Research Article

Synthesis and Some Reactions of 1-aryl-4-acetyl-5-methyl-1,2,3-triazole Derivatives with Anticonvulsant Activity

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 11 Year: 2016 Page: 926-936
Author(s): Ekhlass M. Nassar,Fathy M. Abdelrazek,Rezk R. Ayyad,Ahmed F. El-Farargy

Review Article

Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and Structurally Simplified Analogs. Chemistry and SAR Profile as Adenosine Receptor Antagonists

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 3224-3257
Author(s): Sara Redenti, Antonella Ciancetta, Giorgia Pastorin, Barbara Cacciari, Stefano Moro, Giampiero Spalluto, Stephanie Federico

Mild Synthesis of mono-, bis- and tris 1,2-Dihydrobenzo[4,5]imidazo[1,2- a]pyrimidine Derivatives Using Alkyl Disulfamic Acid Functionalized Magnetic Nanoparticles

Journal: Current Organic Chemistry
Volume: 20 Issue: 1 Year: 2016 Page: 1648-1654
Author(s): Mohammad A. Bodaghifard, Zahra Faraki, Ali R. Karimi

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