Search Result "pyrimidine"


Synthesis and Antimicrobial Activity of New Pyrimidine-Hydrazones

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 1 Year: 2014 Page: 76-81
Author(s): Zafer Asım Kaplancıklı,Leyla Yurttas,Gülhan Turan-Zitouni,Ahmet Özdemir,Gamze Göger,Fatih Demirci,Usama Abu Mohsen

Research Article

Microwave Assisted Synthesis and in vitro Antimicrobial Activities of Fluorine Containing 4-Benzofuran-2-yl-6-phenyl-pyrimidin-2-ylamines

Journal: Medicinal Chemistry
Volume: 10 Issue: 4 Year: 2014 Page: 409-417
Author(s): Tejpal Singh Chundawat,Nutan Sharma,Sunita Bhagat

Facile Synthesis of Novel N4-Substituted 2-(Trifluoromethyl)-tetrahydrobenzothieno[ 2,3-d]pyrimidine Derivatives

Journal: Letters in Organic Chemistry
Volume: 11 Issue: 9 Year: 2014 Page: 700-705
Author(s): Fasong Wang,Hui Gao,Ping Yang,Yan Wang,Xinjian Song

Bu3SnH Assisted Radical Cyclization Towards the Synthesis of Pyrimidine-annulated Spirocyclic and [6,6] Fused Sulfur Heterocycles

Journal: Letters in Organic Chemistry
Volume: 11 Issue: 7 Year: 2014 Page: 487-492
Author(s): K.C. Majumdar, P.K. Maji, S.K. Chattopadhayay

In Silico, Spectroscopic, and Biological Insights on Annelated Pyrrolo[3,2- e]Pyrimidines with Antiproliferative Activity

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 1 Year: 2014 Page: 15-26
Author(s): Antonino Lauria,Alessio Terenzi,Carla Gentile,Annamaria Martorana,Giuseppe Gennaro,Giampaolo Barone,Anna Maria Almerico

In Silico Design of Phenylbenzamide Derivatives Coupled to Pyrimidines as Novel hnRNP K Ligands Against Cancer

Journal: Current Bioactive Compounds
Volume: 10 Issue: 3 Year: 2014 Page: 158-162
Author(s): Matheus G. de Oliveira,Andreza S. Figueredo,Gilberto L.B. de Aquino,Andreia M. Leopoldino,Vinicius B. da Silva,Carlton A. Taft,Carlos H.T. de Paula da Silva

Synthesis and In Vitro Evaluation of Some Hydrazone Derivatives as Potential Antibacterial Agents

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 3 Year: 2014 Page: 355-362
Author(s): Zafer Asim Kaplancikli,Mehlika Dilek Altintop,Ahmet Ozdemir,Gulhan Turan-Zitouni,Gamze Goger,Fatih Demirci

Synthesis, Pharmacological Activity and Molecular Modeling of 1-Aryl-7- hydroxy-2,3-dihydroimidazo[1,2-a]pyrimidine-5(1H)-ones and their 6-Substituted Derivatives

Journal: Medicinal Chemistry
Volume: 10 Issue: 5 Year: 2014 Page: 460-475
Author(s): Marzena Rzadkowska,Elzbieta Szacon,Agnieszka A. Kaczor,Sylwia Fidecka,Ewa Kedzierska,Dariusz Matosiuk

Synthesis of Novel and Highly Functionalized Pyrimidine-5-carboxylate Derivatives and their Antimicrobial Evaluation

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 7 Year: 2014 Page: 930-936
Author(s): Hardik B. Ghodasara, Rajesh G. Vaghasiya, Bharat G. Patel, Viresh H. Shah

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