Search Result "purine-scaffold"


Heterocyclic Scaffolds in the Design of Peptidomimetic Integrin Ligands: Synthetic Strategies, Structural Aspects, and Biological Activity

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2016 Page: 343-359
Author(s): Rossella De Marco,Giacomo Mazzotti,Arianna Greco,Luca Gentilucci

Recent Development in Identification of Potential Novel Therapeutic Targets Against Trypanosomatids

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 20 Year: 2016 Page: 2303-2315
Author(s): Rajender Kumar,Parvati Sharma,Deepak Kumar Gaur,Shikha Jain

Formation of A Novel Purine Metabolite through CYP3A4 Bioactivation and Glutathione Conjugation

Journal: Drug Metabolism Letters
Volume: 10 Issue: 2 Year: 2016 Page: 144-150
Author(s): Julius L. Apuy, Cathie Xiang, Sarah Franc, Sayee G. Hegde, Robert Hubbard, Jingjing Zhao, Mehran F. Moghaddam

Review Article

Design Strategies, Structures and Molecular Interactions of Small Molecule Src Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 8 Year: 2016 Page: 992-1002
Author(s): Sureyya Olgen

Review Article

Microwave Assisted Organic Synthesis of Heterocycles in Aqueous Media: Recent Advances in Medicinal Chemistry

Journal: Medicinal Chemistry
Volume: 12 Issue: 8 Year: 2016 Page: 720-732
Author(s): Francesco Frecentese, Irene Saccone, Giuseppe Caliendo, Angela Corvino, Ferdinando Fiorino, Elisa Magli, Elisa Perissutti, Beatrice Severino, Vincenzo Santagada

2-Arylquinazolin-4(3H)-ones: Inhibitory Activities Against Xanthine Oxidase

Journal: Medicinal Chemistry
Volume: 12 Issue: 1 Year: 2016 Page: 54-62
Author(s): Humaira Zafar,Syed M. Saad,Shahnaz Perveen,Arshia,Rizwana Malik,Ajmal Khan,Khalid M. Khan,Muhammad I. Choudhary

Cytokinin Nucleosides - Natural Compounds with a Unique Spectrum of Biological Activities

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 23 Year: 2016 Page: 2562-2576
Author(s): Mikhail S. Drenichev,Vladimir E. Oslovsky,Sergey N. Mikhailov

Editorial free to download

Editorial (Thematic Issues: New Developments in the Medicinal Chemistry of Some Azoles)

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2016 Page: 3567-3568
Author(s): Nadale K. Downer-Riley, Yvette A. Jackson

Review Article

The Inhibition of Cysteine Proteases Rhodesain and TbCatB: A Valuable Approach to Treat Human African Trypanosomiasis

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2016 Page: 1374-1391
Author(s):

Room Temperature Metal-Free Synthesis of Aryl/Heteroaryl-Substituted Bis(6-aminouracil-5-yl)methanes Using Sulfamic Acid (NH2SO3H) as an Efficient and Eco-friendly Organo-Catalyst

Journal: Current Organocatalysis
Volume: 3 Issue: 2 Year: 2016 Page: 125-132
Author(s): Bubun Banerjee, Goutam Brahmachari

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