Search Result "purine-scaffold"


Research Article

Design and Synthesis of New Substituted Pyrazolopyridines with Potent Antiproliferative Activity

Journal: Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2020 Page: 176-191
Author(s): Vassiliki Giannouli,Nikolaos Lougiakis,Ioannis K. Kostakis,Nicole Pouli,Panagiotis Marakos,Alexios-Leandros Skaltsounis,David A. Horne,Sangkil Nam,Katerina Gioti,Roxane Tenta

Mini-Review Article

Xanthine Scaffold: Available Synthesis Routes to Deliver Diversity by Derivatization

Journal: Mini-Reviews in Organic Chemistry
Volume: 18 Issue: 1 Year: 2021 Page: 27-42
Author(s): Rita Petrucci,Marta Feroci,Leonardo Mattiello,Isabella Chiarotto

Review Article

Thiazolopyrimidine Scaffold as a Promising Nucleus for Developing AnticancerDrugs: A Review Conducted in Last Decade

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 22 Issue: 1 Year: 2022 Page: 2942-2955
Author(s): Md. Rabiul Islam

Research Article

Synthesis, Transformations and Characterization of 8 Aminomethyl Substituted Umbelliferones as Probable Anti-Arrhythmic Agents

Journal: Current Bioactive Compounds
Volume: 15 Issue: 1 Year: 2019 Page: 71-82
Author(s): Alla V. Lipeeva,Arkadiy O. Bryzgalov,Tatyana G. Tolstikova,Elvira E. Shults

Review Article

Multi-Target Directed Ligands (MTDLs): Promising Coumarin Hybrids for Alzheimer’s Disease

Journal: Current Alzheimer Research
Volume: 18 Issue: 1 Year: 2021 Page: 802-830
Author(s): Rohit Bhatia,Sankha S. Chakrabarti,Upinder Kaur,Gaurav Parashar,Anindita Banerjee,Ravindra K. Rawal

Forward Chemical Genetics: Library Scaffold Design

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 7 Issue: 7 Year: 2004 Page: 645-652
Author(s): Sonya M. Khersonsky, Young-Tae Chang

Review Article

Pyrimidine-fused Dinitrogenous Penta-heterocycles as a Privileged Scaf-fold for Anti-Cancer Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 22 Issue: 4 Year: 2022 Page: 284-304
Author(s):

General Review Article

Triazolopyrimidine Nuclei: Privileged Scaffolds for Developing AntiviralAgents with a Proper Pharmacokinetic Profile

Journal: Current Medicinal Chemistry
Volume: 29 Issue: 8 Year: 2022 Page: 1379-1407
Author(s): Tommaso Felicetti,Maria Chiara Pismataro,Violetta Cecchetti,Oriana Tabarrini,Serena Massari

HSP90 Inhibitors: Current Development and Potential in Cancer Therapy

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 9 Issue: 1 Year: 2014 Page: 1-20
Author(s): Katerina Sidera,Evangelia Patsavoudi

An Analysis of the Binding Modes of ATP-Competitive CDK2 Inhibitors as Revealed by X-Ray Structures of Protein-Inhibitor Complexes

Journal: Current Medicinal Chemistry - Anti-Cancer Agents
Volume: 5 Issue: 5 Year: 2005 Page: 561-573
Author(s): A. Vulpetti, P. Pevarello

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