Search Result "novel androstane inhibitors"


Research Article

Steroidal Cardiac Na+/K+ ATPase Inhibitors Exhibit Strong Anti-Cancer Potential in vitro and in Prostate and Lung Cancer Xenografts in vivo

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 14 Issue: 5 Year: 2014 Page: 762-770
Author(s): Konstantinos Dimas, Natalia Papadopoulou, Constantinos Baskakis, Kyriakos C. Prousis, Michail Tsakos, Saad Alkahtani, Sabina Honisch, Florian Lang, Theodora Calogeropoulou, Konstantinos Alevizopoulos, Christos Stournaras

A Steroidal Na+/K+ ATPase Inhibitor Triggers Pro-apoptotic Signaling and Induces Apoptosis in Prostate and Lung Tumor Cells

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 14 Issue: 8 Year: 2014 Page: 1161-1168
Author(s): Sabina Honisch,Saad Alkahtani,Michalis Kounenidakis,Guilai Liu,Saud Alarifi,Hamad Al-Yahya,Konstantinos Dimas,Abdullah A. AlKahtane,Kyriakos C. Prousis,Bader Al-Dahmash,Theodora Calogeropoulou,Konstantinos Alevizopoulos,Florian Lang,Christos Stournaras

Direct and Rapid Transcript Analysis Assay for CYP mRNA Expression and Inducibility in Human Primary Hepatocytes

Journal: Drug Metabolism Letters
Volume: 8 Issue: 2 Year: 2014 Page: 77-87
Author(s): Laura Mattinen,Jenni Kublbeck,Oona Rechardt,Paavo Honkakoski,Jari Rautio

In Vitro Human Hepatocyte-Based Experimental Systems for the Evaluation of Human Drug Metabolism, Drug-Drug Interactions, and Drug Toxicity in Drug Development

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 11 Year: 2014 Page: 1325-1338
Author(s): Albert P. Li

Cytochrome P450s: Mechanisms and Biological Implications in Drug Metabolism and its Interaction with Oxidative Stress

Journal: Current Drug Metabolism
Volume: 15 Issue: 7 Year: 2014 Page: 719-742
Author(s): Sudip Bhattacharyya,Krishnendu Sinha,Parames C. Sil

An Overview of Partial Synthesis and Transformations of Secosteroids

Journal: Current Organic Chemistry
Volume: 18 Issue: 2 Year: 2014 Page: 216-259
Author(s): Katarina Penov Gasi, Marija Sakac, Suzana Jovanovic-Santa, Evgenija Djurendic

Mechanism of Cancer Drug Resistance and the Involvement of Noncoding RNAs

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 26 Year: 2014 Page: 3029-3041
Author(s): Hongping Xia,Kam M. Hui

Role of CNS Transporters in the Pharmacotherapy of HIV-1 Associated Neurological Disorders

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 1 Year: 2014 Page: 1543-1563
Author(s): Tamima Ashraf, Kevin Robillard, Gary N.Y. Chan, Reina Bendayan

Signaling Pathways that Regulate Basal ABC Transporter Activity at the Blood- Brain Barrier

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 1 Year: 2014 Page: 1463-1471
Author(s): David S. Miller, Ronald E. Cannon

Human ABC Transporters at blood-CNS Interfaces as Determinants of CNS Drug Penetration

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 1 Year: 2014 Page: 1450-1462
Author(s):

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