Search Result "nilotinib"


siRNA-Mediated Knock-Down of P-Glycoprotein Expression Reveals Distinct Cellular Disposition of Anticancer Tyrosine Kinases Inhibitors

Journal: Drug Metabolism Letters
Volume: 4 Issue: 2 Year: 2010 Page: 114-119
Author(s): Amina Haouala, Holger Rumpold, Gerold Untergasser, Thierry Buclin, Hans-Beat Ris, Nicolas Widmer, Laurent A. Decosterd

in vitro Anti-leukaemia Activity of Pyrrolo[1,2-b][1,2,5]benzothiadiazepines (PBTDs)

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 5 Issue: 1 Year: 2010 Page: 58-68
Author(s): Gabriella Marfe, Carla Di Stefano

Cardiotoxicity of Tyrosine-Kinase-Targeting Drugs

Journal: Cardiovascular & Hematological Agents in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2010 Page: 11-21
Author(s): A. Garcia-Alvarez, X. Garcia-Albeniz, J. Esteve, M. Rovira, X. Bosch

Gastrointestinal Stromal Tumors: A Paradigm for Therapeutic Options in Solid Organ Tumors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 10 Issue: 7 Year: 2010 Page: 624-634
Author(s): Caroline Novak, Jose G. Trevino

Using Structural and Mechanistic Information to Design Novel Inhibitors/Substrates of P-Glycoprotein

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1769-1774
Author(s): Freya Klepsch, Thomas Stockner, Thomas Erker, Markus Muller, Peter Chiba, Gerhard F. Ecker

The Interactions of Anti-Cancer Drugs Approved in the Last Decade in the United States with Membrane Transporters

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 10 Issue: 8 Year: 2010 Page: 601-616
Author(s): Lokesh Jain, Sophia Abraham, Stacy S. Shord

Influence of Dietary Substances on Intestinal Drug Metabolism and Transport

Journal: Current Drug Metabolism
Volume: 11 Issue: 9 Year: 2010 Page: 778-792
Author(s): Christina S. Won, Nicholas H. Oberlies, Mary F. Paine

Tyrosine Kinase Inhibitors

Journal: Current Cancer Drug Targets
Volume: 10 Issue: 5 Year: 2010 Page: 462-483
Author(s): C. Natoli, B. Perrucci, F. Perrotti, L. Falchi, S. Iacobelli

Hydrophilic Interaction Liquid Chromatography-Tandem Mass Spectrometry for Drug Development

Journal: Current Drug Discovery Technologies
Volume: 7 Issue: 3 Year: 2010 Page: 223-231
Author(s): Andrea L.O.Hebb, Virender Bhan, Alexander D. Wishart, Craig S. Moore, George S. Robertson, Yunsheng Hsieh

Drug-Related Cardiotoxicity for the Treatment of Haematological Malignancies in Elderly

Journal: Current Pharmaceutical Design
Volume: 16 Issue: 2 Year: 2010 Page: 2872-2879
Author(s): Alessandra Malato, Giorgia Saccullo, Giovanni Fazio, Beatrice Vergara, Simona Raso, Giovanni Paolo Guarneri, Antonio Russo, Vincenzo Abbadessa, Sergio Siragusa

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