Search Result "low nanomolar"


Targeting the Plasmepsin 4 Orthologs of Plasmodium sp. with “Double Drug” Inhibitors

Journal: Protein & Peptide Letters
Volume: 15 Issue: 9 Year: 2008 Page: 868-873
Author(s): Linda Janka, Jose Clemente, N. Vaiana, A. Sparatore, Sergio Romeo, Ben M. Dunn

Novel RGD Peptidomimetics Embedding 1,2,3-Triazole as Central Scaffold; Synthesis and αvβ3 Integrin Affinity

Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 5 Year: 2011 Page: 401-405
Author(s): Ming Hong Ni, Emiliano Esposito, Massimo Castorina, Alma Dal Pozzo

General Research Article

Design and Synthesis of New JAK1 Inhibitors based on Sulfonamide-Triazine Conjugates

Journal: Current Computer-Aided Drug Design
Volume: 17 Issue: 7 Year: 2021 Page: 916-926
Author(s): Safa Daoud,Mutasem O. Taha

First Discovery of Tylophora Alkaloids as HIV Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 12 Issue: 4 Year: 2015 Page: 277-283
Author(s): Ziwen Wang,Mingxiao Wang,Lei Wang,Xue Yao,Yue Li,Juan Tan,Wentao Qiao,Yunqi Geng,Yuxiu Liu,Qingmin Wang

Dangerous Liaisons between Beta-Amyloid and Cholinergic Neurotransmission

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 1 Year: 2014 Page: 2525-2538
Author(s): Stefano Govoni, Elisa Mura, Stefania Preda, Marco Racchi, Cristina Lanni, Massimo Grilli, Stefania Zappettini, Alessia Salamone, Guendalina Olivero, Anna Pittaluga, Mario Marchi

Low Molecular Weight Compounds with Transition Metals as Free Radical Scavengers and Novel Therapeutic Agents

Journal: Cardiovascular & Hematological Agents in Medicinal Chemistry
Volume: 8 Issue: 3 Year: 2010 Page: 128-146
Author(s): Andrea Bencini, Paola Failli, Barbara Valtancoli, Daniele Bani

Dual Cyclooxygenase and Carbonic Anhydrase Inhibition by Nonsteroidal Anti-Inflammatory Drugs for the Treatment of Cancer

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 24 Year: 2015 Page: 2812-2818
Author(s): Celeste De Monte,Simone Carradori,Andrea Gentili,Adriano Mollica,Daniela Trisciuoglio,Claudiu T. Supuran

Low Molecular Weight Inhibitors of the Protease Anthrax Lethal Factor

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 8 Issue: 3 Year: 2008 Page: 290-306
Author(s): Georgios A. Spyroulias, Georgios A. Dalkas, Athanasios Papakyriakou, Alexios Vlamis-Gardikas

Advances in Matrix Metalloproteinase Inhibitors Based on Pyrrolidine Scaffold

Journal: Current Medicinal Chemistry
Volume: 15 Issue: 4 Year: 2008 Page: 374-385
Author(s): Wen-Fang Xu, Xian-Chao Cheng, Qiang Wang, Hao Fang

Review Article

Carbon Paste Modified Electrode as Powerful Sensor Approach Determination of Food Contaminants, Drug Ingredients, and Environmental Pollutants: A Review

Journal: Current Analytical Chemistry
Volume: 15 Issue: 4 Year: 2019 Page: 410-422
Author(s): Hassan Karimi-Maleh,Fatemeh Karimi,Morteza Rezapour,Majede Bijad,Mohammad Farsi,Aliasghar Beheshti,Seyed-Ahmad Shahidi

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