Search Result "lead optimization"


Computer-Aided Drug Design: Lead Discovery and Optimization

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 15 Issue: 4 Year: 2012 Page: 328-337
Author(s): Mingli Xiang, Yu Cao, Wenjie Fan, Lijuan Chen, Yirong Mo

Back to the Future: Lessons Learned in Modern Target-based and Whole-Cell Lead Optimization of Antimalarials

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2012 Page: 473-483
Author(s): Arnab K. Chatterjee, Bryan K.S. Yeung

Vibration Characteristic Analysis and Collaborative Optimization Design for the Disk Brake

Journal: Recent Patents on Mechanical Engineering
Volume: 5 Issue: 3 Year: 2012 Page: 220-226
Author(s): Fangwei Xie,Gang Zheng,Hewei Wang,Xiuwen Yang,Yanfang Zhao

Multi-Parameter Optimization: Identifying High Quality Compounds with a Balance of Properties

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 9 Year: 2012 Page: 1292-1310
Author(s): Matthew D. Segall

Applications of Biophysical Tools to Target-Based Discovery of Novel Antibacterial Leads

Journal: Current Drug Targets
Volume: 13 Issue: 3 Year: 2012 Page: 388-408
Author(s): Sushmita Lahiri, Steven Kazmirski, Gunther Kern, Gautam Sanyal

Optimization of fructooligosaccharides synthesis by immobilized fructosyltransferase

Journal: Current Chemical Biology
Volume: 6 Issue: 1 Year: 2012 Page: 42-52
Author(s): Elizama Aguiar-Oliveira,Maria Isabel Rodrigues,Francisco Maugeri

History, Principle and Techniques for Waveform Optimization in External Defibrillations

Journal: Recent Patents on Engineering
Volume: 6 Issue: 1 Year: 2012 Page: 20-30
Author(s): Changlin Yin, Bihua Chen, Lei Gao, Yongqin Li

Portfolio Optimization: New Challenges and Perspectives

Journal: Recent Patents on Computer Science
Volume: 5 Issue: 1 Year: 2012 Page: 59-65
Author(s): Marina Resta

Prediction of Optimal pH and Temperature of Cellulases Using Neural Network

Journal: Protein & Peptide Letters
Volume: 19 Issue: 1 Year: 2012 Page: 29-39
Author(s): Shao-Min Yan, Guang Wu

Multi-Objective Optimization Methods in De Novo Drug Design

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 10 Year: 2012 Page: 979-987
Author(s): C. A. Nicolaou,C. Kannas,E. Loizidou

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