Search Result "lead optimization"


Advances in the Integration of Drug Metabolism into the Lead Optimization Paradigm

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 6 Year: 2009 Page: 703-716
Author(s): Walter A. Korfmacher

Methodologies to Assess Brain Drug Delivery in Lead Optimization

Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2009 Page: 148-162
Author(s): Margareta Hammarlund-Udenaes, Ulf Bredberg, Markus Friden

Methods for Integrating and Handling Complex Optimization Problems in the Process Industries

Journal: Recent Patents on Chemical Engineering
Volume: 2 Issue: 2 Year: 2009 Page: 123-127
Author(s): Edwin Zondervan, Andre B. de Haan

From Fragment Screening to Potent Binders: Strategies for Fragment-to-Lead Evolution

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 8 Year: 2009 Page: 956-961
Author(s): Krystian Eitner, Uwe Koch

Early Toxicity Screening and Selection of Lead Compounds for Parasitic Diseases

Journal: Current Drug Targets
Volume: 10 Issue: 3 Year: 2009 Page: 291-298
Author(s): Renata Campos Nogueira, Jose Fernando Oliveira-Costa, Matheus Santos de Sa, Ricardo Ribeiro dos Santos, Milena Botelho Pereira Soares

Research Development on (KxNa1-x)NbO3-Based Lead-Free Piezoelectric Ceramics

Journal: Recent Patents on Materials Science
Volume: 2 Issue: 2 Year: 2009 Page: 140-153
Author(s): Jiagang Wu, Dingquan Xiao, Jianguo Zhu

Fragment Library Screening and Lead Characterization Using SPR Biosensors

Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2009 Page: 1725-1735
Author(s): U. Helena Danielson

Potential Factors Induced by Filoviruses that Lead to Immune Supression

Journal: Current Molecular Medicine
Volume: 9 Issue: 2 Year: 2009 Page: 174-185
Author(s): Mansour Mohamadzadeh

Design, Optimization, Preparation and Evaluation of Dispersion Granules of Valsartan and Formulation into Tablets

Journal: Current Drug Delivery
Volume: 6 Issue: 1 Year: 2009 Page: 28-37
Author(s): Agnivesh R. Shrivastava, Bhalchandra Ursekar, Chhanda J. Kapadia

Chinese Grain Production Forecasting Method Based on Particle Swarm Optimization-based Support Vector Machine

Journal: Recent Patents on Engineering
Volume: 3 Issue: 1 Year: 2009 Page: 8-12
Author(s): Sheng-Wei Fei, Yu-Bin Miao, Cheng-Liang Liu

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