Search Result "kinase inhibitor"


Review Article

Heteroaromatic Pim Kinase Inhibitors Containing a Pyrazole Moiety

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 11 Issue: 3 Year: 2016 Page: 309-321
Author(s): Pascale Moreau,Fabrice Anizon,Francis Giraud,Yannick J. Esvan

ROS1 Kinase Inhibitors for Molecular-Targeted Therapies

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 2 Year: 2016 Page: 142-160
Author(s): M.M. Al-Sanea,A.Z. Abdelazem,B.S. Park,K.H. Yoo,T. Sim,Y.J. Kwon,S.H. Lee

Old Tyrosine Kinase Inhibitors and Newcomers in Gastrointestinal Cancer Treatment

Journal: Current Cancer Drug Targets
Volume: 16 Issue: 2 Year: 2016 Page: 175-185
Author(s): Erika Giordani,Federica Zoratto,Martina Strudel,Anselmo Papa,Luigi Rossi,Marina Minozzi,Davide Caruso,Eleonora Zaccarelli,Monica Verrico,Silverio Tomao

Benzofuran Small Molecules as Potential Inhibitors of Human Protein Kinases. A Review

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 7 Year: 2016 Page: 879-894
Author(s): Halina Kwiecień,Agata Goszczyńska,Paulina Rokosz

In silico Modeling of Antimalarial Protein Kinase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 2 Year: 2016 Page: 129-134
Author(s): Rahul Balasaheb Aher,Kunal Roy

Review Article

Mutant B-Raf Kinase Inhibitors as Anticancer Agents

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 12 Year: 2016 Page: 1558-1575
Author(s): Vivek Asati,Sanjay K. Bharti,Debarshi K. Mahapatra

Review Article

Cell Cycle Kinases in Osteosarcoma: Potential for Therapeutic Intervention

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 3 Year: 2016 Page: 4830-4834
Author(s): Li Cheng, Chongchong Wang, Juehua Jing

Studies on the IC50 of Trisubstituted Thiazoles as Cdc7 Kinase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 1 Year: 2016 Page: 33-42
Author(s): Huazhen Yang,Xun Liu,Zhiling Ye,Fucheng Song,Lianhua Cui,Zhuang Yu,Hongzong Si,Honglin Zhai

Anaplastic Lymphoma Kinase Inhibitors in Non-Small Cell Lung Cancer

Journal: Current Drug Targets
Volume: 17 Issue: 6 Year: 2016 Page: 739-745
Author(s): David M. Straughan, Sa d C. Azoury, Vivek Shukla

Review Article

Exploring Pyrimidine Pharmacophore as Thymidine Monophosphate Kinase Inhibitors for Antitubercular Activity: A Review

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 3211-3223
Author(s): Trupti Sameer Chitre, Kalyani Dhirendra Asgaonkar, Shital Manoj Patil, Muthu Kumaradoss Kathiravan, Subhash Balkrishna Padhye

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