Search Result "inverse agonists"


Histamine H3 Receptor (H3R) Antagonists and Inverse Agonists in the Treatment of Sleep Disorders

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 1 Year: 2011 Page: 1426-1429
Author(s): Meredith Broderick, Tony Masri

The Evolution of Histamine H3 Antagonists/Inverse Agonists

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 6 Year: 2011 Page: 648-660
Author(s): Evan P. Lebois, Carrie K. Jones, Craig W. Lindsley

GABAA Receptor Subtype-Selective Modulators. II. α5-Selective Inverse Agonists for Cognition Enhancement

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 9 Year: 2011 Page: 1203-1214
Author(s): John R. Atack

Glutamate Receptor Agonists: Stereochemical Aspects

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 7 Year: 2011 Page: 887-906
Author(s): Stine Byskov Vogensen, Jeremy R. Greenwood, Lennart Bunch, Rasmus Praetorius Clausen

Pharmacophore and 3D-QSAR Studies on 1-Sulfonyl-4-acylpiperazines as Selective Cannabinoid-1 Receptor (CB1R) Inverse Agonists

Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 7 Year: 2011 Page: 659-670
Author(s): Vikas N. Telvekar, Lalit B. Thakur, Prashant B. Jagdhane, Yogesh D. Manohar

Latest Advances Towards the Discovery of 5-HT7 Receptor Ligands

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1108-1121
Author(s): V. Pittala, D. Pittala

Molecular Determinants of Selective Agonist and Antagonist Binding to the Histamine H4 Receptor

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 6 Year: 2011 Page: 661-679
Author(s): Enade P. Istyastono, Chris de Graaf, Iwan J.P. de Esch, Rob Leurs

High-Density Lipoprotein Cholesterol-Elevating Effect of a Novel Peroxisome Proliferator-Activated Receptor δ Agonist

Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 6 Year: 2011 Page: 496-499
Author(s): Shogo Sakuma, Tsuyoshi Endo, Takashi Kanda, Hideki Nakamura, Satomi Yamasaki, Tomio Yamakawa

Obesity and Gastrointestinal Hormones-Dual Effect of Angiotensin II Receptor Blockade and a Partial Agonist of PPAR-γ

Journal: Current Vascular Pharmacology
Volume: 9 Issue: 2 Year: 2011 Page: 162-166
Author(s): Hironori Nakagami, Ryuichi Morishita

A Pharmacological Primer of Biased Agonism

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 92-98
Author(s): Bradley T. Andresen

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