Search Result "inverse agonist"


Review Article

Design and Synthesis of Dopaminergic Agonists

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 2 Year: 2016 Page: 2790-2825
Author(s): Maria Soledad Matute, Rosa Matute, Pedro Merino

Antineoplastic Effects of PPAR? Agonists, with a Special Focus on Thyroid Cancer

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 7 Year: 2016 Page: 636-649
Author(s): Silvia Martina Ferrari, Gabriele Materazzi, Enke Baldini, Salvatore Ulisse, Paolo Miccoli, Alessandro Antonelli, Poupak Fallahi

Review Article

Hemopressin Peptides as Modulators of the Endocannabinoid System and their Potential Applications as Therapeutic Tools

Journal: Protein & Peptide Letters
Volume: 23 Issue: 12 Year: 2016 Page: 1045-1051
Author(s): Giorgia Macedonio,Azzurra Stefanucci,Cristina Maccallini,Sako Mirzaie,Ettore Novellino,Adriano Mollica

Research Article

Relationship Between Susceptibility to DMCM-Induced Generalized Motor Convulsions and Low-Affinity [3H]-Ouabain Binding in Membranes in Rat Brain

Journal: Current Molecular Pharmacology
Volume: 9 Issue: 4 Year: 2016 Page: 332-336
Author(s): Marcos Brandao Contó,Marco Antonio Campana Venditti

Research Article

Gut Microbiota of Obese, Type 2 Diabetic Individuals is Enriched in Faecalibacterium prausnitzii, Akkermansia muciniphila and Peptostreptococcus anaerobius after Weight Loss

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 16 Issue: 2 Year: 2016 Page: 99-106
Author(s): Marlene Remely, Berit Hippe, Julia Zanner, Eva Aumueller, Helmuth Brath, Alexander G. Haslberger

Immunotherapy and Hormone-therapy in Metastatic Breast Cancer: A Review and an Update

Journal: Current Drug Targets
Volume: 17 Issue: 10 Year: 2016 Page: 1127-1139
Author(s): Andrea Nicolini,Angelo Carpi,Paola Ferrari,Pier Mario Biava,Giuseppe Rossi

Novel Therapeutic Targets for Management of Type-2 Diabetes Mellitus

Journal: Immunology, Endocrine & Metabolic Agents in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2016 Page: 18-30
Author(s): Anishkumar Chaurasia, Rashmi Mallya, Tabassum Khan

Review Article

A Systematic Review and Meta-Analysis of Controlled Trials on the Effects of Statin and Fibrate Therapies on Plasma Homocysteine Levels

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 39 Year: 2016 Page: 4490-4503
Author(s): Amirhossein Sahebkar,Matteo Pirro,Željko Reiner,Arrigo Cicero,Gianna Ferretti,Mario Simental-Mendía,Luis E. Simental-Mendía

Effect of Dipeptidyl Peptidase-4 Inhibitors on Plasma Adiponectin: A Systematic Review and Meta-Analysis of Randomized Controlled Trials

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 13 Year: 2016 Page: 1356-1369
Author(s): Amirhossein Sahebkar,Valentina Ponzo,Simona Bo

Review Article open access plus

Classification of Therapeutic and Experimental Drugs for Brown Adipose Tissue Activation: Potential Treatment Strategies for Diabetes and Obesity

Journal: Current Diabetes Reviews
Volume: 12 Issue: 4 Year: 2016 Page: 414-428
Author(s): Jogeshwar Mukherjee, Aparna Baranwal, Kimberly N. Schade

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