Search Result "inverse agonist"


Atypical antipsychotics and inverse agonism at 5-HT2 receptors

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 26 Year: 2015 Page: 3732-3738
Author(s): Laura C. Sullivan,William P Clarke,Kelly A. Berg

Research Article

Synthetic Cannabinoid Receptor Agonists and Antagonists: Implication in CNS Disorders

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 10 Issue: 2 Year: 2015 Page: 142-156
Author(s): Clementina Manera, Chiara Arena, Andrea Chicca

When is a Proof-of-Concept (POC) not a POC? Pomaglumetad (LY2140023) as a Case Study for Antipsychotic Efficacy

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 26 Year: 2015 Page: 3788-3796
Author(s): Gerard J. Marek

Research Article

Peptide Agonists and Antagonists with Potential Application in Neurological Disorders

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 10 Issue: 2 Year: 2015 Page: 76-89
Author(s): Anna Russo, Sara La Manna, Giancarlo Morelli, Ettore Novellino, Daniela Marasco

Do Histamine receptor 3 antagonists have a place in the therapy for schizophrenia?

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 26 Year: 2015 Page: 3760-3770
Author(s): Bart A. Ellenbroek,Bibinaz Ghiabi

Research Article

Phytocannabinoids and Cannabimimetic Drugs: Recent Patents in Central Nervous System Disorders

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 10 Issue: 2 Year: 2015 Page: 157-177
Author(s): Roberta Ranieri, Daniela Marasco, Maurizio Bifulco, Anna M. Malfitano

Direct Estimation of CaV1.2 Gating Parameters: Quantification of Voltage Sensor – Pore Transductions and their Modulation by FLP 64176

Journal: Current Molecular Pharmacology
Volume: 8 Issue: 1 Year: 2015 Page: 87-94
Author(s): Beyl Stanislav,Kügler Philipp,Timin Eugen,Hering Steffen

Structure Diversity, Synthesis, and Biological Activity of Cyathane Diterpenoids in Higher Fungi

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 19 Year: 2015 Page: 2375-2391
Author(s): Hao-Yu Tang,Xia Yin,Cheng-Chen Zhang,Qian Jia,Jin-Ming Gao

Classical Neurotransmitters and Neuropeptides Involved in Parkinson's Disease: Focus on Anti-Parkinsonian Drugs

Journal: Current Drug Therapy
Volume: 10 Issue: 2 Year: 2015 Page: 66-81
Author(s): Felix-Martin Werner,Rafael Coveñas

Discovery of GPCR Ligands by Molecular Docking Screening: Novel Opportunities Provided by Crystal Structures

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 24 Year: 2015 Page: 2484-2503
Author(s): David Rodríguez,Anirudh Ranganathan,Jens Carlsson

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