Search Result "integrase strand transfer inhibitors"


Research Article

Computational Studies of N-substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors using 3D-QSAR, Pharmacophore Modeling and Molecular Docking

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 11 Year: 2017 Page: 1291-1302
Author(s): Yuming Luo,Yujie Ren,Xiaodong Gao

Research Article

Integrase Strand Transfer Inhibitors and the Emergence of Immune Reconstitution Inflammatory Syndrome (IRIS)

Journal: Current HIV Research
Volume: 15 Issue: 6 Year: 2017 Page: 405-410
Author(s): Mina Psichogiou,Dimitrios Basoulis,Maria Tsikala-Vafea,Stefanos Vlachos,Christos J. Kapelios,Georgios L. Daikos

Review Article

Recent Advances in Antiretroviral Agents: Potent Integrase Inhibitors

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 18 Year: 2017 Page: 2552-2567
Author(s): Mina Psichogiou,Garyphalia Poulakou,Dimitrios Basoulis,Dimitrios Paraskevis,Antonios Markogiannakis,George L. Daikos

Review Article

Novel Second Generation HIV Integrase Inhibitor-DOLUTEGRAVIR: An Emerging Weapon Against HIV

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 3 Year: 2017 Page: 354-371
Author(s): Vivek Jain,Diksha Gupta,Ashutosh Pareek,Yashumati Ratan

Research Article

Quantitative Structure-Activity Relationship and Docking Studies on a Series of Oxadiazole and Triazole Substituted Naphthyridines as HIV-1 Integrase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 10-27
Author(s): Basheerulla Shaik,Vijay Agrawal,Satya P. Gupta,Urvana Menon

Research Article

Molecular Docking and Molecular Dynamics Simulation Based Approach to Explore the Dual Inhibitor Against HIV-1 Reverse Transcriptase and Integrase

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 8 Year: 2017 Page: 734-746
Author(s): Subhash Chander,Rajan Kumar Pandey,Ashok Penta,Bhanwar Singh Choudhary,Manish Sharma,Ruchi Malik,Vijay Kumar Prajapati,Sankaranarayanan Murugesan

Research Article

HIV Type 1 Integrase Natural Polymorphisms in Viral Variants Circulating in FSU Countries

Journal: Current HIV Research
Volume: 15 Issue: 5 Year: 2017 Page: 318-326
Author(s): Ilya Lapovok,Vita Laga,Elena Kazennova,Marina Bobkova

Review Article

Applying Knowledge of Enzyme Biochemistry to the Prediction of Functional Sites for Aiding Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 21 Year: 2017 Page: 2401-2421
Author(s): Priyadarshini P. Pai,Sukanta Mondal

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Journal: Current Organic Synthesis
Volume: 14 Issue: 6 Year: 2017 Page: 755-755
Author(s): Terrence R. Burke

Research Article

An Improved Preparation of (R)-3-Aminobutanol, a Key Intermediate for the Synthesis of Dolutegravir Sodium

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 1371-1375
Author(s): Y. Srinivasa Rao, B. Hari Babu, I. Aminual, D. Nageshwar , P.V.V. Satyanarayana

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